Review on Biological Activities of 1,3,4-Thiadiazole Derivatives

Arvind k. Singh, Geeta Mishra, Kshitiz Jyoti

Pages: 44-49

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Design, Characterization and Biological Activity of a new series of s-Triazines Derived with Morpholine

Kalpesh S. Parikh, Sandip P. Vyas

DOI: 10.7324/JAPS.2012.2519Pages: 111-114

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Estimation of Naratriptan Hydrochloride in Bulk and Formulation by First Order Derivative UV-Spectrophotometric Methods

Jayshri S. Borse, Atul A. Shirkhedkar

DOI: 10.7324/JAPS.2012.2642Pages: 227-229

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Biological activities of [1,2,4] triazolo-[3,4-b],[1,3,4]-thiadiazole-6-yl) (o-tolyamino) methylazetidin-2-one

Harcharan Lal, Neeraj Sharma, T.P. Agarwal and Nitin Sharma

DOI: 10.7324/JAPS.2012.21021Pages: 104-112

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Derivative Spectrophotometric Methods for the Determination of Zolpidem Tartrate in Tablets

M. Mathrusri Annapurna, B. Swathi, M. Siri Chandra and K. Tulasi

DOI: 10.7324/JAPS.2012.21117Pages: 096-099

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A Validated Comparitative LC and Ratio First Derivative Spectrophotometric Method for the Simultaneous Determination of Levocetrizine dihydrochloride and Montelukast sodium in Bulk and Pharmaceutical dosage forms

R. Swethan Babu, K. Anirudha Bharadwaj, N.C Arjun, Nagaraj, Venkatesh Prasad

DOI: 10.7324/JAPS.2012.2842Pages: 243-249

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Solid Dispersion: Methods and Polymers to increase the solubility of poorly soluble drugs

Ladan Akbarpour Nikghalb, Gurinder Singh, Gaurav Singh and Kimia Fazaeli Kahkeshan

DOI: 10.7324/JAPS.2012.21031Pages: 170-175

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Analytical method development and validation of sitagliptine phosphate monohydrate in pure and tablet dosage form by derivative spectroscopy

G. Jeyabalan and Narendra Nyola

DOI: 10.7324/JAPS.2013.30118Pages: 095-098

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Scopoletin, a coumarin derivative compound isolated from Macaranga gigantifolia Merr

Akhmad Darmawan, Soleh Kosela, Leonardus B.S. Kardono, and Yana M. Syah

DOI: 10.7324/JAPS.2012. 21231Pages: 175-177

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Spectrophotometric Methods for Determination of Tapentadol Hydrochloride

Mokhtar M. Mobrouk, Hamed M. El-Fatatry, Sherin F. Hammad, Aya A. Mohamed

DOI: 10.7324/JAPS.2013.30324Pages: 122-125

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Molecular docking study of 3,6 bis(3’substituted propoxy) and 3,6 bis (5’substituted pentyloxy) xanthone derivatives as PGHS- 2 inhibitors

Aparoop Das, Pratap Parida, Neha Agarwal, Jaya shree, Brajesh Shankar and Dipankar Chakraborty

DOI: 10.7324/JAPS.2013.34.S3Pages: S13-S22

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Binding affinity of asiatic acid derivatives design against Inducible Nitric Oxide Synthase and ADMET Prediction

RE Kartasasmita, I Musfiroh, A Muhtadi, S Ibrahim

DOI: 10.7324/JAPS.2014.40213Pages: 075-080

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Simple Spectrophotometric and HPTLC-Densitometric Methods for Determination of Cefdinir in Bulk Powder and Pharmaceuticals, and in Presence of its Hydrolytic Degradation Products

Omar Abdel-Aziz, Maha Farouk, Reham Nagi, Laila Abdel-Fattah

DOI: 10.7324/JAPS.2014.40722Pages: 129-136

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Design, synthesis, molecular docking of new thiopyrimidine-5-carbonitrile derivatives and their cytotoxic activity against HepG2 cell line

Ahmad F. Eweas, Qasem M.A. Abdallah, Emad S.I. Hassan

DOI: 10.7324/JAPS.2014.41218Pages: 102-111

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Environmental biotoxicity screening of some pyrrole and 1,4-dihydropyridine heterocyclic derivatives

A. Idhayadhulla, Aseer Manilal, Behailu Merdekios and R. Surendra Kumar

DOI: 10.7324/JAPS.2015.50519Pages: 101-105

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Synthesis of barbituric acid derivatives using microwave irradiation method and in vitro evaluation of antimicrobial and cytotoxic activity

M. A. Sattar, Mst. Khodeza Khatun, Rafiquel Islam, Md. Hossain Sohrab, Sharif M. Al-Reza

DOI: 10.7324/JAPS.2015.501106Pages: 038-042

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Recent Advances and Future Prospects of Phthalimide Derivatives

Neelottama Kushwaha, Darpan Kaushik

DOI: 10.7324/JAPS.2016.60330Pages: 159-171

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Pyrimidinethione derivatives with tosyl substitution: Synthesis, and antimicrobial property investigation

Shubhalaxmi, B. S. Manjunatha, K. Ananda, K. Subrahmanya Bhat

DOI: 10.7324/JAPS.2016.60613Pages: 073-078

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Antioxidant Properties and Phytochemical Contents of Garcinia schomburgkiana Pierre.

Imron Meechai, Worrapong Phupong, Warangkana Chunglok, Puttinan Meepowpan

DOI: 10.7324/JAPS.2016.60618Pages: 102-107

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Simultaneous estimation of Aliskiren hemifumarate and Hydrochlorothiazide in combined Tablet Formulation by Simultaneous equation, Absorbance ratio and First derivative Spectroscopic Methods

Ashim Kumar Sen, Dhanya B Sen, Rajesh A Maheshwari, Ramachandran Balaraman, Avinash K Seth

DOI: 10.7324/JAPS.2016.60724Pages: 164-170

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Analytical method development and validation for simultaneous estimation of Teneligliptin hydrobromide hydrate and Metformin hydrochloride from it’s pharmaceutical dosage form by three different UV spectrophotometric methods

Ashim Kumar Sen, Denish N. Hinsu, Dhanya B. Sen, Aarti S. Zanwar, Rajesh A. Maheshwari, Vikas R. Chandrakar

DOI: 10.7324/JAPS.2016.60924Pages: 157-165

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QSAR and Molecular Docking of Phthalazine Derivatives as Epidermal Growth Factor Receptor (EGFR) Inhibitors

Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2017.70427Pages: 181-191

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Design, Synthesis and Preliminary Pharmacological Screening (antimicrobial, analgesic and anti-inflammatory activity) of Some Novel Quinazoline Derivatives

Biswajit Dash, Suvakanta Dash, Damiki Laloo, Chitrani Medhi

DOI: 10.7324/JAPS.2017.70612Pages: 083-096

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Synthesis, Pharmacological Evaluation, Molecular Docking and in silico ADMET Prediction of Nitric Oxide Releasing Biphenyls as Anti-Inflammatory Agents

Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2017.71006Pages: 037-047

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Docking Evaluation of Catechin and its Derivatives on Fat Mass and Obesity-Associated (FTO) Protein for Anti-Obesity Agent

Tony Sumaryada, Renti Efraim Marimpola Simamora, Laksmi Ambarsari

DOI: 10.7324/JAPS.2018.8810Pages: 063-068

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The employment of spectroscopic techniques coupled with chemometrics for authentication analysis of halal pharmaceuticals

Abdul Rohman, Nina Salamah

DOI: 10.7324/JAPS.2018.81009Pages: 063-068

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3D-QSAR analysis of pyrimidine derivatives as AXL kinase inhibitors as anticancer agents

Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2018.81103Pages: 015-027

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Synthesis and anticancer potential of aminomethyl derivatives of methyl-substituted asymmetrical curcumin mono-carbonyl

Arini Kurnia, Fadlina Chany Saputri, Hayun Hayun

DOI: 10.7324/JAPS.2019.90803Pages: 018-024

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Comparison of UV-spectrophotometric and RP-HPLC methods for estimation of deflazacort in solid dosage form

Manisha Puranik, Samta Shambharkar, Shantanu Nimbalkar, Debarshi Kar Mahapatra

DOI: 10.7324/JAPS.2020.10711Pages: 082-088

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Development and validation of two spectrophotometric methods for simultaneous determination of diosmine and hesperidin in mixture and their applications

Ismail Bennani, Madiha Alami Chentoufi, Ibrahim Sbai El Otmani, Amine Cheikh, Nouriddin Bamou, Miloud El Karbane, Mustapha Bouatia

DOI: 10.7324/JAPS.2020.10713Pages: 100-107

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New benzimidazole derivatives as inhibitors of Pteridine reductase 1: Design, molecular docking study and ADMET prediction

Shraddha Phadke, Rakesh Somani, Devender Pathak

DOI: 10.7324/JAPS.2020.10904Pages: 030-039

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Design, synthesis, and evaluation of some novel N-benzothiazol-2-yl benzamide derivatives as allosteric activators of human glucokinase

Sandeep Arora, Ajmer Singh Grewal, Neelam Sharma, Kunal Arora, Ervon Dhalio, Sukhbir Singh

DOI: 10.7324/JAPS.2021.11s104Pages: 038-047

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Design, synthesis and in silico prediction of drug-likeness properties of new ortho, meta and para-(2-cyano-3-(3,5-di-tert-butyl-4- hydroxyphenyl)acrylamido)benzoic acids

Madhavi Kuchana, Lakshmi Bhavani Kambala

DOI: 10.7324/JAPS.2021.110805Pages: 031-035

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Evaluating the effect of amine-geldanamycin hybrids on anticancer activity

Tipparat Samsawat, Chanjira Jaramornburapong, Weerachai Phutdhawong, Waya S. Phutdhawong, Thongchai Taechowisan

DOI: 10.7324/JAPS.2021.110814Pages: 098-107

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Antioxidant potential and LC/MS metabolic profile of anticancer fractions from Echium angustifolium Mill. aerial parts

Hanan M. El-Tantawy, Ahmed R. Hassan, Hala E. Taha

DOI: 10.7324/JAPS.2021.1101220Pages: 200–208

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Synthesis and evaluation of novel 4-anilinocoumarin derivatives as potential antimicrobial agents

Sonia Yadav, Nitin Kumar, Vijay Bhalla

DOI: 10.7324/JAPS.2022.120518Pages: 196-204

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In silico and in vitro anti-cancer activity against breast cancer cell line MCF-7 of amide cinnamate derivatives

Teni Ernawati, Nina Artanti, Yudhi Dwi Kurniawan

DOI: 10.7324/JAPS.2024.162177Pages: 102-107

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Synthesis, in-vitro antioxidant and anti-inflammatory properties of novel amide derivatives of substituted 2-aminothiophenes and 3,4-dimethoxy cinnamic acid

Satya Sree Bandaru, Madhavi Kuchana

DOI: 10.7324/JAPS.2024.180925Pages: 116-125

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