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February, 2019

Volume: 9, Issue: 2

In this Issue: Research Article: 14, Short Communication: 5

19 Feb, 2019   Research Article

Antitumor activities of new iso(thio)cyanates and their nitrogen and sulphur heterocyclic phosphorus derivatives

Mansoura A. Abd-El-Maksoud, Aida I. El-Makawy, Sekena H. Abdel-Aziem, Soher S. Maigali, Marwa El-Hussieny, Shaimaa T. Mansour, Fouad M. Soliman

DOI: 10.7324/JAPS.2019.90201Pages: 001-011

21 Feb, 2019   Research Article

Synthesis and anticonvulsant activity of 6-methyl-2-thioxo-2, 3-dihydropyrimidin-4(1H)-one acetamides

Hanna Severina, Olha Skupa, Andrei Khairulin, Natalya Voloshchuk, Victoria Georgiyants

DOI: 10.7324/JAPS.2019.90202Pages: 012-019

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21 Feb, 2019   Research Article

In silico predictive for modification of chalcone with pyrazole derivatives as a novel therapeutic compound for targeted breast cancer treatment

Riska Prasetiawati, Adel Zamri, Melisa Intan Barliana, Muchtaridi Muchtaridi

DOI: 10.7324/JAPS.2019.90203Pages: 020-028

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19 Feb, 2019   Research Article

A validated LC-MS/MS method for the pharmacokinetic study of alogliptin in healthy rabbits

Yatha Ravi, Bigala B. Rajkamal

DOI: 10.7324/JAPS.2019.90204Pages: 029-037

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19 Feb, 2019   Research Article

Antiproliferative and apoptosis inducing potential of whole plant extracts of Sesuvium portulacastrum against different cancer cell lines

Sathvika Chintalapani, M. S. Swathi, Mangamoori Lakshmi Narasu

DOI: 10.7324/JAPS.2019.90205Pages: 038-043

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21 Feb, 2019   Research Article

A descriptive cross-sectional study to evaluate the Generic Drug User Fee Act: A boon or loss to the Indian generic pharmaceutical industry

Sarika Prasanna Pardhe

DOI: 10.7324/JAPS.2019.90206Pages: 044-051

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21 Feb, 2019   Research Article

Recycling of expired paracetamol-containing drugs as source of useful reagents for an organic synthesis

Inna Puzanova, Andrii Lozynskyi, Lilia Lesyk, Bohdan Hromovyk, Roman Lesyk

DOI: 10.7324/JAPS.2019.90207Pages: 052-056

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19 Feb, 2019   Research Article

Treatment patterns of antipsychotics and clinical features for treating patients with schizophrenia at the teaching hospital in Jakarta, Indonesia

Wawaimuli Arozal, Diana Wijaya, Vivaian Soetikno, Nurmiati Amir, Rianto Setiabudy

DOI: 10.7324/JAPS.2019.90208Pages: 057-063

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19 Feb, 2019   Research Article

Biological activity of Passiflora edulis f. Flavicarpa ethanolic leaves extract on human colonic adenocarcinoma cells

Valentina Ramirez, Sandra Sulay Arango, Maria Elena Maldonado, Diego Uribe, Johanny Aguillon, Jenny Paola Quintero, Nelsy Loango

DOI: 10.7324/JAPS.2019.90209Pages: 064-071

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21 Feb, 2019   Research Article

Phytochemical compounds of anise hyssop (Agastache foeniculum) and antibacterial, antioxidant, and acetylcholinesterase inhibitory properties of its essential oil

Ivan G. Ivanov, Radka Z. Vrancheva, Nadezhda T. Petkova, Yulian Tumbarski, Ivayla N. Dincheva, Ilian K. Badjakov

DOI: 10.7324/JAPS.2019.90210Pages: 072-078

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22 Feb, 2019   Research Article

RP-HPLC method for determination of norethindrone in dissolution media and application to study release from a controlled release nanoparticulate liquid medicated formulation

Suhair S. Al-Nimry, Bashar M. Altaani, Razan H. Haddad

DOI: 10.7324/JAPS.2019.90211Pages: 079-086

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22 Feb, 2019   Research Article

Studying activity and toxicity of different TNF-alpha inhibitors in controlling patients with active ulcerative colitis

Bahir Abdul Razzaq Mshimesh

DOI: 10.7324/JAPS.2019.90212Pages: 087-096

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25 Feb, 2019   Research Article

A post-market quality assessment of first-line, fixed-dose combination antiretrovirals in South Africa

Kim Ward, Reem Suleiman, Yunus Kippie, Admire Dube

DOI: 10.7324/JAPS.2019.90213Pages: 097-104

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25 Feb, 2019   Research Article

Evaluation of Cissus populnea gum as a directly compressible matrix system for tramadol hydrochloride extended-release tablet

Olutayo Ademola Adeleye, Mbang N. Femi-Oyewo, Michael A. Odeniyi, Tolulope O. Ajala

DOI: 10.7324/JAPS.2019.90214Pages: 105-111

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25 Feb, 2019   Short Communication

A simplified system for simulation of Streptococcus mutans biofilm on healthy extracted human tooth as dental plaque model

Nadia Halib, Nor Zaihana Abdul Rahman, Rohazila Mohamad Hanafiah, Nabihah Roslan, Nurhani Jauhar

DOI: 10.7324/JAPS.2019.90215Pages: 112-115

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25 Feb, 2019   Short Communication

Spectroscopic identification of brominated, non-brominated alkaloids and evaluation of antimicrobial activity of Eudistomin-I, Eudistomin H, from green ascidian Eudistoma viride

Rajaian Pushpabai Rajesh, Annappan Murugan

DOI: 10.7324/JAPS.2019.90216Pages: 116-123

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25 Feb, 2019   Short Communication

Qualitative anti-tubercular activity of synthetic ethyl 7-acetyl2-substituted-3-(4-substituted benzoyl) indolizine-1-carboxylate analogues

Sandeep Chandrashekharappa, Katharigatta N. Venugopala, Rashmi Venugopala, Basavaraj Padmashali

DOI: 10.7324/JAPS.2019.90217Pages: 124-128

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25 Feb, 2019   Short Communication

Distribution and antimicrobial activity of Thai marine actinomycetes

Wongsakorn Phongsopitanun, Khanit Suwanborirux, Somboon Tanasupawat

DOI: 10.7324/JAPS.2019.90218Pages: 129-134

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25 Feb, 2019   Short Communication

Scientific research presentations in pharmacoeconomics and health outcomes research: status of India compared to SAARC and BRICS countries

Sreeranjani Menon, Harshith Nayak, Virendra Ligade

DOI: 10.7324/JAPS.2019.90219Pages: 135-140

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