Review on Biological Activities of 1,3,4-Thiadiazole Derivatives

Arvind k. Singh, Geeta Mishra, Kshitiz Jyoti

Pages: 44-49

Graphical Abstract

Epigenetic modification of suppressor of cytokine signaling-3 in asthmatic mouse lung: role of interleukin-6

Vani Mishra, Rahul Sharma, Brajadulal Chattopadhyay, Bhola Nath Paul

Pages: 81-89

Graphical Abstract

Synthesis and in-vitro screening of 3,4-dihydropyrimidin-2(1H)-one derivatives for antihypertensive and calcium channel blocking activity

Hiren M. Marvaniya, Palak K. Parikh, Dhrubo Jyoti Sen

Pages: 109-113

Graphical Abstract

Synthesis, characterization and anti-trypanosomal activity of R-(-)carvone and arylketones-thiosemi carbazones and toxicity against Artemia salina Leach

Bienvenu Glinma, Salome D. S. Kpoviessi, Raymond H. Fatondji, Fernand A. Gbaguidi, Coco N. Kapanda, Joanne Bero, Didier M. Lambert, Veronique Hannaert, Joëlle Quetin-Leclercq, Mansourou Moudachirou, Jacques Poupaert, Georges C. Accrombessi

Pages: 65-70

Graphical Abstract

Enhancement of camptothecin production in Camptotheca acuminata hairy roots by overexpressing ORCA3 gene

Xiaoning Ni, Shiqiu Wen, Wei Wang, Xiaoyun Wang, Hui Xu, Guoyin Kai

Pages: 85-88

Graphical Abstract

Antifungal activity of bioactive compound of seeds of Psoralea corylifolia L. against seed borne Fusarium species of maize

Kiran. B, Lalitha.V, Raveesha.K.A

Pages: 161-164

Graphical Abstract

Histological Studies in Murine Model of Asthma: Effect of Stat3 siRNA

Bhushan Chaudhari, Pankaj Jagdale, Sheikh Raisuddin, Shambhoo Sharan Tripathi, Mamta Shukla, Pradeep Kumar Singh, Pradeep Kumar

Pages: 77-84

Graphical Abstract

Gastro-Retentive Floating Matrix Tablets of Cefpodoxime Proxetil

K. Sreenivasa Rao, Rakesh R. Vairagkar, Dattatreya B. Udgirkar, Praveen S. Patil, Karnakumar V. Biradar

Pages: 190-194

Graphical Abstract

Improving Oral Bioavailability of Agaricoglycerides by Solid Lipid-Based Self-Emulsifying Drug Delivery System

Chun Chao Han, Linna Han

Pages: 195-199

Graphical Abstract

Antihyperlipidaemic Activity of Spermacoce Hispida Ethanolic Extract in Triton WR-1339 Induced Hyperlipidaemic Rats

G. Sivaelango, P. Senthil Kumaran, P. Kumaravel, P. Revathi, A. Jaswant

Pages: 95-98

Graphical Abstract

Genotoxicity of anticancer drug Azathioprine (Imuran): role of Omega-3 (?-3) oil as protective agent

Elelaimy I.A, Elfiky S.A., Hassan A.M., Ibrahim H.M., Elsayad R.I.

DOI: 10.7324/JAPS.2012.2404Pages: 14-23

Graphical Abstract

Community Pharmacy/Hospital Based Assessment of Clinical Pharmacist Intervention for Safe and Effective Drug Use

Awofisayo Sunday Olajide, Aboyarin Oladayo, Udoh Imo Emmanuel

DOI: 10.7324/JAPS.2012.2424Pages: 66-69

Graphical Abstract

GC-MS analysis of Polygala rosmarinifolia Wights & Arn

M. Alagammal, P. Tresina Soris, V.R. Mohan

DOI: 10.7324/JAPS.2012.2504Pages: 188-190

Graphical Abstract

In-Vitro Anthelmintic Activity of Croton Bonplandianum Baill

Hapse S.A., Pagar H.J. Suruse S.D., Ugale S.S.

DOI: 10.7324/JAPS.2012.2516Pages: 191-193

Graphical Abstract

Comparative in vitro antibacterial activities study of some mucoadhesive polymeric suspensions containing fluoroquinolones

Chandra Kanti Chakraborti, Subhashree Sahoo, Pradipta Kumar Behera, Anjulata Manjari Sahoo

DOI: 10.7324/JAPS.2012.2502Pages: 44-48

Graphical Abstract

Simultaneous determination of pioglitazone and glimepiride in their pharmaceutical formulations

Mamdouh R. Rezk, Safa'a M. Riad, Ghada Y. Mahmoud, Abdel-Aziz El Bayoumi Abdel Aleem

DOI: 10.7324/JAPS.2012.2544Pages: 177-184

Graphical Abstract

Synthesis and antimicrobial activity of novel (3,5-dichloro-4-((5-aryl-1,3,4-thiadiazol-2-yl)methoxy) phenyl) aryl methanones

V. Srinivasa Murthy, B. K. Manuprasad, S. Shashikanth

DOI: 10.7324/JAPS.2012.2726Pages: 172-176

Graphical Abstract

Chemical Constituents of the Essential Oil of Laggera pterodonta (DC.) Sch. Bip. From North-Central Nigeria

Egharevba Henry Omoregie, Kunle Folashade Oluyemisi, Okwute Simon Koma, Okogun Joseph Ibumeh

DOI: 10.7324/JAPS.2012.2835Pages: 198-202

Graphical Abstract

Isolation of a novel triterpene from the Essential oil of fresh leaves of Chromolaena odorata and its in-vitro cytotoxic activity against HepG2 cancer cell line

Velliangiri Prabhu and Subban Ravi

DOI: 10.7324/JAPS.2012.2926Pages: 132-136

Graphical Abstract

Synthesis of novel Naphthalene COX inhibitors for anti-inflammatory activity

Anand B. Pandya, Dhaval G. Prajapati, Saurabh S. Pandya

DOI: 10.7324/JAPS.2012.2840Pages: 226-232

Graphical Abstract

HPLC evaluation on 3-n-butylphthalide distribution

Qi Wang, Shuoyang Li, Peifeng Liu, Ming Shen, Tao Gong, Yourong Duan, Zhang Zhi-Rong

DOI: 10.7324/JAPS.2012.21003Pages: 016-020

Graphical Abstract

Anti-ischemic effect of ethyl acetate extract of Aquilaria crassna by attenuation of p38-MAPK activation

Chanyatip Suwannasing, Nitchawat Paiyabhroma, Sarawut Kumphune

DOI: 10.7324/JAPS.2012.21005Pages: 026-030

Graphical Abstract

Three component one pot synthesis of 5-Substituted 1-Aryl-2,3-diphenyl imidazoles: A novel class of promising antioxidants

Nagaraja Naik, H. Vijay Kumar, J. Rangaswamy, S.T. Harinia and T.C. Umeshkumar

DOI: 10.7324/JAPS.2012.21112Pages: 067-074

Graphical Abstract

3',4'-Dimethoxy Quercetin, a Flavonol Compound Isolated from Kalanchoe pinnata

Akhmad Darmawan, Megawati and Sofa Fajriah

DOI: 10.7324/JAPS.2013.30116Pages: 088-090

Graphical Abstract

Synthesis and Antihypertensive Activity of Some Quinazoline Derivatives

Harsha U. Patel, Ravi S. Patel, Chhaganbhai N. Patel

DOI: 10.7324/JAPS. 2013.30332Pages: 171-174

Graphical Abstract

Study of Complex Nutrients, Temperature and Salts on Hyaluronic acid Production In Streptococcus zooepidermicus ATCC 43079

Nguyen Tu Hoang Khue and Pham Thien Minh Vo

DOI: 10.7324/JAPS.2013.3503Pages: 012-015

Graphical Abstract

Formulation and In-Vitro Characterization of Acyclovir Floating Matrix Tablets: A Factorial Design Study

Sadhana Shahi, Ashok Sonawane, Suhas Vanamore, Nityanand Zadbuke

DOI: 10.7324/JAPS.2013.3513Pages: 065-074

Graphical Abstract

Possible Involvement of 'Phosphatidylinositol-3 kinase and endothelial nitric oxide synthase' in experimental obesity induced vascular endothelium dysfunction

Gargee Dubey, PL Sharma and Saurabh Sharma

DOI: 10.7324/JAPS.2013.3608Pages: 052-060

Graphical Abstract

Glypican-3 as a tumor marker for hepatocellular carcinoma

Amal A. Mohamed, Naglaa El-Toukhy, M. Magdi Atta, Salah M. Ahmed

DOI: 10.7324/JAPS.2013.3613Pages: 083-087

Graphical Abstract

Exopolysaccharide in Lactobacillus Rhamnosus Pn04 After Co-Culture with Leuconostoc mesenteroides Vtcc-B-643

Nguyen Tu Hoang Khue and Nguyen Huu Ngoc

DOI: 10.7324/JAPS.2013.3703Pages: 014-017

Graphical Abstract

Measuring Interesting Amino Acid Patterns for Alzheimer's Disease Related Studies Targets on the Binding Site Using Association Rule Mining

D. Ponmary Pushpa Latha and D. Joseph Pushpa Raj

DOI: 10.7324/JAPS.2013.3705Pages: 025-030

Graphical Abstract

Determination of Total Arsenic in Indonesian Tuna Fish Sample

Tiny A. Koesmawati, B. Buchari, Muhammad B. Amran, Leonardus B.S. Kardono

DOI: 10.7324/JAPS.2013.3722Pages: 116-121

Graphical Abstract

Microwave assisted synthesis of 3-α-carboxy ethylrhodanine derivatives and their in vitro antibacterial activity

Kaveri Sundaram and Subban Ravi

DOI: 10.7324/JAPS.2013.3725Pages: 133-135

Graphical Abstract

Enteric coating of hard gelatin capsules by the spouted bed process

H.V.A. Oliveira, M.P.G. Peixoto, L.A. Tacon & L.A.P.Freitas

DOI: 10.7324/JAPS.2013.3810Pages: 057-063

Graphical Abstract

Statistical Optimization of Olanzapine Ternary Solid Dispersions with Pvp K 30 and Peg 20,000 by Response Surface Methodology

Anil Katharia, Ratendra Kumar, Rajiv Sharma, Yogendra Singh, Uday Veer Singh Teotia

DOI: 10.7324/JAPS.2013.3920Pages: 109-116

Graphical Abstract

In silico Analysis of 3D-QSAR and Molecular Docking for Bcl-2 Inhibitors to Potential Anticancer Drug Development

Ramachandran M, Balwin Nambikkairaj, Kumaran K, Arun Kumar De and G.Ramesh Kumar

DOI: 10.7324/JAPS.2013.31005Pages: 023-029

Graphical Abstract

Efficacy of 5-(2-aroyl)aryloxy methyl-2-phenyl-1,3,4-oxadiazoles as antibacterial and antifungal agents

Bushra Begum A, Noor Fatima Khanum, Naveen P, Lakshmi Ranganatha V, Asha MS and Shaukath Ara Khanum

DOI: 10.7324/JAPS.2013.31119Pages: 105-109

Graphical Abstract

Cytotoxic effects of antiglypican-3 against HepG2 cell line

Randa A Zaghloul, Mohammed M H Al-Gayyar, Mamdouh M El-Shishtawy, Mohamed A. Ebrahim

DOI: 10.7324/JAPS.2013.31206Pages: 031-035

Graphical Abstract

3D QSAR and Pharmacophore Modelling on Chalcones as Antileishmanial Agents potential Trypanothione reductase Inhibitors

Sujit Arun Desai, Santosh Sahedeo Kumbhar, Vishal Shankar Katti, Prafulla Balkrishna Choudhari, Manish Sudesh Bhatia

DOI: 10.7324/JAPS.2013.31218Pages: 099-102

Graphical Abstract

Computational analysis of phytocompounds with 1,3-β-D-Glucan synthase for antidermatophytic activity

M Jeyam, M Arangaraj, P Ravikumar, G Shalini

DOI: 10.7324/JAPS.2014.40211Pages: 064-069

Graphical Abstract

Synthesis of Methyl 2-Cinnamamido-3-Hydroxy Propanoate Having Activity against P388 Leukemia Cells

Teni Ernawati, Yulia Anita, Puspa Dewi Lotulung and Muhammad Hanafi

DOI: 10.7324/JAPS.2014.40318Pages: 092-095

Graphical Abstract

Effect of formulation parameters on Sumatriptan succinate Buccal Mucoadhesive Tablet: Quality by Design approach

Wable Arti J, Thokal Seema B, Mittal Sandeep S, Shirsat Ajinath E, Bhingare Chandrashekhar L, Ingle Pramod L

DOI: 10.7324/JAPS.2014.40418Pages: 103-111

Graphical Abstract

In vitro cytotoxicity effects of single and combination Nigella sativa and Zingiber zerumbet extracts on human myeloid leukemia (HL60) cells and its mode of cell death

Norfazlina M.N., Farida Zuraina M.Y., Rajab N.F, Mohd Nazip S., Rumiza A.R., Suziana Zaila C.F., Lek Mun L., Nurshahirah N., Florinsiah L.

DOI: 10.7324/JAPS.2014.40509Pages: 051-055

Graphical Abstract

Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines

Guillaume Burgy, Emmanuelle Limanton, François Carreaux, Emilie Durieu, Laurent Meijer, and Jean-Pierre Bazureau

DOI: 10.7324/JAPS.2014.40604Pages: 025-032

Graphical Abstract

Cytotoxic activity and apoptosis induction of 8-hydroxyisocapnolactone-2´,3´-diol and its combination with Doxorubicin on MCF-7 and T47D cells

Ratna Asmah Susidarti, Riris Istighfari Jenie, Muthi’ Ikawati, Dyaningtyas Dewi Pamungkas Putri, Edy Meiyanto

DOI: 10.7324/JAPS.2014.40614Pages: 089-097

Graphical Abstract

Piceatanol: Anti-Cancer Compound From Gewang Seed Extract

Leny Heliawati, Agus Kardinan, Tri Mayanti, Roekmi-ati Tjokronegoro

DOI: 10.7324/JAPS.2015.50119Pages: 110-113

Graphical Abstract

Evaluation as antioxidant agents of 1,2,4-triazole derivatives: effects of essential functional groups

Ahmet Cetin, Ibrahim Halil Geçibesler

DOI: 10.7324/JAPS.2015.50620Pages: 120-126

Graphical Abstract

Formulation and in vitro evaluation of berberine containing liposome optimized by 32 full factorial designs

Girish Sailor, A K Seth, Ghanshyam Parmar, Sachin Chauhan, Ankur Javia

DOI: 10.7324/JAPS.2015.50704Pages: 023-028

Graphical Abstract

Chemical Constituents of Cordia dichotoma G. Forst.

Consolacion Y. Ragasa, Virgilio Ebajo Jr., Mariquit M. De Los Reyes, Emelina H. Mandia, Maria Carmen S. Tan, Robert Brkljača, Sylvia Urban

DOI: 10.7324/JAPS.2015.58.S3Pages: 016-021

Graphical Abstract

Chemical constituents of Cycas aenigma

Vincent Antonio S. Ng, Esperanza Maribel G. Agoo, Chien-Chang Shen, Consolacion Y. Ragasa

DOI: 10.7324/JAPS.2015.50906Pages: 032-036

Graphical Abstract

Synthesis and screening of new maleimide derivatives as potential anti-tubercular agents

Saroj Kumar Sahoo, Kurre Purna Nagasree, Jamullamudi Risy Namratha, Pemmadi Raghuveer Varma, Muthyala Murali Krishna Kumar

DOI: 10.7324/JAPS.2015.510.S8Pages: 044-047

Graphical Abstract

In silico analysis of indole-3-carbinol and its metabolite DIM as EGFR tyrosine kinase inhibitors in platinum resistant ovarian cancer vis a vis ADME/T property analysis

Raju Dash, S. M. Zahid Hosen, Md. Rezaul Karim, Mohammad Shah Hafez Kabir, Mohammed Munawar Hossain, Md. Junaid, Ashekul Islam, Arkajyoti Paul, Mohammad Arfad Khan

DOI: 10.7324/JAPS.2015.501112Pages: 073-078

Graphical Abstract

Pharmacokinetics interaction of dapoxetine with different doses of green tea extract in male healthy volunteers using midazolam as CYP3A4 enzyme probe

Khaled Sobhy Abdelkawy, Ahmed M Donia, Mahmoud S Abdallah

DOI: 10.7324/JAPS.2015.501201Pages: 001-007

Graphical Abstract

Cytotoxic effect and apoptotic activity of Parmentiera edulis DC. hexane extract on the breast cancer cell line MDA-MB-231

Cynthia Carolina Estanislao Gómez, Cynthia Ordaz Pichardo, Eduardo San Martín Martínez, Nury Pérez Hernández, Guillermo Pérez Ishiwara, María del Consuelo Gómez García

DOI: 10.7324/JAPS.2016.600103Pages: 015-022

Graphical Abstract

Synthesis, Evaluation and Docking Study of 1, 3, 5-Triazine Derivatives as Cytotoxic Agents against Lung Cancer

Marwa F. Balaha, Mervat H. El-Hamamsy, Nabawya A. Sharaf El-Din, Nageh A.El-Mahdy

DOI: 10.7324/JAPS.2016.60405Pages: 028-045

Graphical Abstract

Synthesis and antibacterial activity of novel 2-(arylimino)thiazolidin-4-one and 2-(benzylidenehydrazono)-3-arylthiazolidin-4-one derivatives

Ebaa M. El-Hossary, Yassin M. Nissan, Katharina Edkins, Heike Bruhn

DOI: 10.7324/JAPS.2016.60502Pages: 007-017

Graphical Abstract

Production of antioxidant xylooligosaccharides from lignocellulosic materials using Bacillus amyloliquifaciens NRRL B-14393 xylanase

Mona M. Rashad, Abeer E. Mahmoud, Mohamed U. Nooman, Hadeer A. Mahmoud, Alaa El-Din M.M. El-Torky, Akaber T. Keshta

DOI: 10.7324/JAPS.2016.60606Pages: 030-036

Graphical Abstract

A preliminary evaluation of anticancer and antioxidant potential of two traditional medicinal plants from Lamiaceae-Pogostemon heyneanus and Plectranthus amboinicus

Vaishali Rai, Vinitha Ramanath Pai, Pratapchandra Kedilaya

DOI: 10.7324/JAPS.2016.60811Pages: 073-078

Graphical Abstract

Mechanism of Relaxant Action of Ethyl 6-amino-5-cyano-2-methyl- 4-(pyridin-4-yl)-4H-pyran-3-carboxylate Mainly Through Calcium Channel Blockade in Isolated Rat Trachea

Soledad Alemán-Pantitlán, César Millán-Pacheco, Miguel A. Vázquez, Fernando Hernández-Borja, Rafael Villalobos-Molina, Blanca Bazán-Perkins, Samuel Estrada-Soto

DOI: 10.7324/JAPS.2016.601004Pages: 029-036

Graphical Abstract

Synthesis, spectroscopic characterization and biological applications of Cu(II) and Ni(II) complexes with 2-butyl-4-chloro-5-formylimidazole thiosemicarbazone

A. Sreenath Reddy, L. Sivarama Krishna, H. K. Rashmi, P. Uma Maheswari Devi, Y. Sarala, A. Varada Reddy

DOI: 10.7324/JAPS.2016.601015Pages: 107-112

Graphical Abstract

Clonazepam associated hypothyroidism: Aforethought on a concealed dilemma

Rupam Gill, Dipanjan Bhattacharjee, Navin A. Patil, Shripathy M. Bhat

DOI: 10.7324/JAPS.2016.601031Pages: 222-225

Graphical Abstract

Antifeedant Constituents from Leucaena leucocephala

Poonam Negi, Bhupendra Singh Rawat, Devendra Singh Negi

DOI: 10.7324/JAPS.2016.601204Pages: 028-031

Graphical Abstract

Effect of intensive endurance training on rat brain and hepatic 8-oxoguanine DNA glycosylase and 8-hydroxy-2'-deoxyguanosine levels

Mohammad Esmaiel Afzalpour, Hossein TaheriChadorneshin, Seyed-Hosein Abtahi-Eivary, Ehsan Afroozi-Gerow

DOI: 10.7324/JAPS.2016.601215Pages: 110-113

Graphical Abstract

Nanochemopreventive effect of polymer functionalized gold nanoparticles containing hesperetin drug inhibited proliferation and induced apoptosis in Hep3B cells

Gokuladhas Krishnan, Jayakumar Subramaniyan, Pramila Chengalvarayan Subramani, Devaki Thiruvengadam

DOI: 10.7324/JAPS.2016.601216Pages: 114-123

Graphical Abstract

Effect of exogenous application of indole-3-acetic acid (IAA) on cell maturity of Olea europaea L. and extractability of phenolic compounds in virgin olive oil

Youssef MOUSTAKIME, Zakaria HAZZOUMI, Zain El Abidine FATEMI, Khalid AMRANI JOUTEI

DOI: 10.7324/JAPS.2017.70228Pages: 199-206

Graphical Abstract

QSAR and Molecular Docking of Phthalazine Derivatives as Epidermal Growth Factor Receptor (EGFR) Inhibitors

Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2017.70427Pages: 181-191

Graphical Abstract

Synthesis and evaluation of silver nanoparticles using Cymodocea rotundata against clinical pathogens and human osteosarcoma cell line

Jayanthi Abraham, Shantanu Saraf, Vakas Mustafa, Yugal Chaudhary, Silambarasan Sivanangam

DOI: 10.7324/JAPS.2017.70608Pages: 055-061

Graphical Abstract

Synthesis and antimicrobial activity of Bis-Derivatives of 3a′, 6a′Dihydro-2'H-Spiro[Indole-3,1'-Pyrrolo[3,4-c]Pyrrole]-2,4',6'(1H, 3'H, 5'H)-Trione

Ruslan Gr. Redkin, Evgeniya I. Syumka, Leonid A. Shemchuk, Valentin P. Chernykh

DOI: 10.7324/JAPS.2017.70610Pages: 069-078

Graphical Abstract

Design, Synthesis and Preliminary Pharmacological Screening (antimicrobial, analgesic and anti-inflammatory activity) of Some Novel Quinazoline Derivatives

Biswajit Dash, Suvakanta Dash, Damiki Laloo, Chitrani Medhi

DOI: 10.7324/JAPS.2017.70612Pages: 083-096

Graphical Abstract

Evaluation of Plant Food Extracts in Experimental Model of Alzheimer's Like Disease Induced by Aluminum Lactate in Rats

Sahar Y. Al-Okbi, Doha A. Mohamed, Mohamed Abdel Fatah, Kholoud Abdel Aal, Shaimaa E Mohammed

DOI: 10.7324/JAPS.2017.70712Pages: 070-076

Graphical Abstract

Computational, structural and functional aspects of hypothetical protein of Aspergillus flavus Pheromone Receptor Pre-A (PRP-A)

Maneesh Kumar, Sindhuprava Rana, Harish Kumar, Pratik Kumar, Manas Ranjan Dikhit, Rani Mansuri, Jainendra Kumar, Ganesh Chandra Sahoo

DOI: 10.7324/JAPS.2017.70714Pages: 089-097

Graphical Abstract

Synthesis and establishment of Amlodipine impurity G reference standard

Ly Dieu Ha, Trang Thi Diem Nguyen, Tri Minh Le

DOI: 10.7324/JAPS.2017.71015Pages: 105-110

Graphical Abstract

Anticancer Activity of New Substituted Pyrimidines, Their Thioglycosides and Thiazolopyrimidine Derivatives

Mahmoud N. M. Yousif, Wael A. El-Sayed, Hebat-Allah S. Abbas, Hanem M. Awad, Nabil M. Yousif

DOI: 10.7324/JAPS.2017.71104Pages: 021-032

Graphical Abstract

Steroids and isoquercetin from Lygodium microphyllum

Hadi Kuncoro, Kindi Farabi, Laode Rijai

DOI: 10.7324/JAPS.2017.71120Pages: 136-141

Graphical Abstract

QSAR, Molecular Docking and Dynamics Studies of Pyrrolo[2,3-b]Pyridine Derivatives as Bruton’s Tyrosine Kinase Inhibitors

Ruslin, Nirwana, Muhammad Arba, Mukhsar, Daryono Hadi Tjahjono

DOI: 10.7324/JAPS.2017.71201Pages: 001-007

Graphical Abstract

Accessing the Anti-Proliferating Activity of Tankyrase-2 Inhibitors via 2D, 3D-QSAR and Molecular Docking: Assessment of Structure Activity Relationships

Mervat H. El-Hamamsy

DOI: 10.7324/JAPS.2017.71203Pages: 014-027

Graphical Abstract

Quality of Life Assessment in Cancer Patients of Regional Centre of Hyderabad City

V. Naga Sunanda M. Priyanka, J. Architha1 , M. Shravan, A. Srinivasa Rao, Mohd. Abdul Hadi

DOI: 10.7324/JAPS.2018.8125Pages: 165-169

Graphical Abstract

Anti-inflammatory and antioxidant activity of salicylic acid conjugated dihydropyrazoline analogues

Naveen Puttaswamy, Rekha N D, Lakshmi Ranganatha V, Prashanth T, Shaukath Ara Khanum

DOI: 10.7324/JAPS.2018.8209Pages: 060-064

Graphical Abstract

Alkaline Phosphatase Activity of Marsilea crenata Presl. Extract and Fractions as Marker of MC3T3-E1 Osteoblast Cell Differentiation

Burhan Ma’arif, Mangestuti Agil, Hening Laswati

DOI: 10.7324/JAPS.2018.8308Pages: 55-59

Graphical Abstract

Computational Model of Doxorubicin Conjugate with Docosahexaenoic Acid and Integrin αvβ3 Ligand for Anticancer

Ace T. Hidayat, Muhammad Yusuf, Husein H. Bachti, Ajeng Diantini, Achmad Zainuddin

DOI: 10.7324/JAPS.2018.8401Pages: 001-006

Graphical Abstract

Cisplatin-Induced Nephrotoxicity in Rats: Modulatory Role of Simvastatin and Rosuvastatin against Apoptosis and Inflammation

Rasha E. Mostafa, Dalia O. Saleh, Dina F. Mansour

DOI: 10.7324/JAPS.2018.8406Pages: 043-050

Graphical Abstract

Molecular Docking Studies Involving the Inhibitory Effect of Gymnemic Acid, Trigonelline and Ferulic Acid, the Phytochemicals with Antidiabetic Properties, on Glycogen Synthase Kinase 3 (α and β)

V. Roshana Devi, C. Sharmila, S. Subramanian

DOI: 10.7324/JAPS.2018.8422Pages: 150-160

Graphical Abstract

QSAR, Molecular Docking and Dynamics Studies of Quinazoline Derivatives as Inhibitor of Phosphatidylinositol 3-Kinase

Muhammad Arba, Ruslin, Waode Umi Kalsum, Armid Alroem, Muhammad Zakir Muzakkar, Ida Usman, Daryono Hadi Tjahjono

DOI: 10.7324/JAPS.2018.8501Pages: 001-009

Graphical Abstract

Synthesis and Evaluation of Antimitotic Activity of N-Phenyl Tetralones

Umesha Basavaiah, Sowbhagya, Vinaya, Yeriyur Basavaiah Basavaraju

DOI: 10.7324/JAPS.2018.8512Pages: 094-100

Graphical Abstract

Design, One-pot Synthesis and Biological Evaluation of Imidazo[2,1-b] [1,3,4] Thiadiazole Derivatives for their Anti- Tubercular and Anti-Fungal Activity

Manjoor Ahamad Syed, Yiragam Reddy Padmanabha Reddy, K. B. Chandrasekhar

DOI: 10.7324/JAPS.2018.8704Pages: 021-027

Graphical Abstract

Effect of Kirganelia reticulata extract on Human Embryonic Kidney cells with evidence on morphological changes

Madhurima Ghosh, Jhinuk Chatterjee, V. Krishnamurthy

DOI: 10.7324/JAPS.2018.8917Pages: 114-118

Graphical Abstract

3D-QSAR analysis of pyrimidine derivatives as AXL kinase inhibitors as anticancer agents

Siddharth J. Modi, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2018.81103Pages: 015-027

Graphical Abstract

Effects of sea urchin (Diadema setosum) gonad extracts on gene expression of FOXP3 and the production of cytokine on Salmonella typhi-induced mice

Wa Ode Salma, Sitti Wahyuni, Nursin Kadir, Suryani Asad, Irawan Yusuf 

DOI: 10.7324/JAPS.2018.81216Pages: 140-146

Graphical Abstract

In silico evaluation of Benzo (f) chromen-3-one as a potential inhibitor of NF-κB: A key regulatory molecule in inflammation-mediated pathogenesis of diabetes, Alzheimer’s, and cancer

Sandeep Kumar Gandham, Venkata Ramaiah Chintha, Rajendra Wudayagiri

DOI: 10.7324/JAPS.2018.81218Pages: 157-164

Graphical Abstract

3D-QSAR, molecular docking, and dynamics simulation of quinazoline–phosphoramidate mustard conjugates as EGFR inhibitor

Ruslin Ruslin, Resky Amelia, Yamin Yamin, Sandra Megantara, Chun Wu, Muhammad Arba

DOI: 10.7324/JAPS.2019.90113Pages: 089-097

Graphical Abstract

In silico predictive for modification of chalcone with pyrazole derivatives as a novel therapeutic compound for targeted breast cancer treatment

Riska Prasetiawati, Adel Zamri, Melisa Intan Barliana, Muchtaridi Muchtaridi

DOI: 10.7324/JAPS.2019.90203Pages: 020-028

Graphical Abstract

Qualitative anti-tubercular activity of synthetic ethyl 7-acetyl2-substituted-3-(4-substituted benzoyl) indolizine-1-carboxylate analogues

Sandeep Chandrashekharappa, Katharigatta N. Venugopala, Rashmi Venugopala, Basavaraj Padmashali

DOI: 10.7324/JAPS.2019.90217Pages: 124-128

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Anti-diabetic drug, metformin, and the p38 inhibitor (SB203580) reduces internal organs oxidative stress in non-obese type 2 diabetic rats

Nuttikarn Nokkaew, Jantira Sanit, Podsawee Mongkolpathumrat, Siyamon Boontawee, Supanut Ithipruchyabun, Wannapa Plangklang, Punyanuch Adulyaritthikul, Kantapich Kongpol, Sarawut Kumphune

DOI: 10.7324/JAPS.2019.90502Pages: 012-020

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3D-QSAR, molecular docking and dynamics simulation of difluorophenol pyridine derivatives as RSK2 inhibitor

Muhammad Arba, Hamzah Azali, Sabarudin Ombe, Alrum Armid, Ida Usman

DOI: 10.7324/JAPS.2019.90601Pages: 001-009

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15N-NMR spectroscopic studies and investigation of spectral data property relationships of proton pump inhibitors

Bhanumathi Devi NC, Someswara Rao N., Tamal Ghosh, Alok Mukerjee

DOI: 10.7324/JAPS.2019.90608Pages: 061-066

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Identification of polyketide synthase 13 inhibitor: Pharmacophore-based virtual screening and molecular dynamics simulation

Muhammad Arba, Andy-Nur Hidayat, Henny Kasmawati, Yamin Yamin, Ida Usman

DOI: 10.7324/JAPS.2019.90702Pages: 012-017

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The effect of metformin and P38 MAPK inhibitor on diabetic bone porosity in non-obese type 2 diabetic rats

Punyanuch Adulyaritthikul, Jantira Sanit, Nuttikarn Nokkaew, Kantapich Kongpol, Podsawee Mongkolpathumrat, Sakarat na Lampang, Catleya Rojviriya, Sarawut Kumphune

DOI: 10.7324/JAPS.2019.90711Pages: 082-090

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Isolation of flavonol rhamnosides from Pometia pinnata leaves and investigation of α-glucosidase inhibitory activity of flavonol derivatives

Fadhila Utari, Afrizal Itam, Syafrizayanti Syafrizayanti, Widya Hasvini Putri, Masayuki Ninomiya, Mamoru Koketsu, Kaori Tanaka, Mai Efdi

DOI: 10.7324/JAPS.2019.90808Pages: 053-065

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Synthesis, in-vitro antioxidant activity and in-silico prediction of drug-likeness properties of a novel compound: 4-(3,5-Di-tert-butyl- 4-hydroxybenzylidene)-3-methylisoxazol-5(4H)-one

Madhavi Kuchana, Durga Rani Bethapudi, Ragini Katamarajugari Ediga, Yoshitha Sisapuram

DOI: 10.7324/JAPS.2019.90915Pages: 105-110

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Synthesis, characterization, and in vitro release of oxytetracycline loaded in pH-responsive CaCO3 nanoparticles

Sherifat Banke Idris, Arifah Abdul Kadir, Faez Firdaus Abdullah Jesse, Siti Zubaidah Ramanoon, Muhammad Abdul Basit, Zainul Amiruddin Zakaria, Md Zuki Abu Bakar Zakaria

DOI: 10.7324/JAPS.2019.91103Pages: 019-027

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Believes versus evidence-based regio-orientation in the structure assignment of pyrazolo[1,5-a]pyrimidines

Mosaad Sayed Mohamed, Asmaa Mahmoud Mahmoud

DOI: 10.7324/JAPS.2019.91117Pages: 126-144

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Pharmacokinetic drug–drug interaction study between clindamycin and cyclosporin in rabbits

Issam Mohammed Abushammala, Lama Attef El Gussein, Badea Elzaman Zomlot, Kamal Fakher Abushammalleh, Mohammed Mahmoud Taha, Mohammed Yousef Miqdad

DOI: 10.7324/JAPS.2020.102016Pages: 108-111

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Isolation, characterization, and cytotoxic studies of secondary metabolites from the leaves of Bauhinia foveolata Dalzell: An endemic tree from the Western Ghats, India

Prasanna V. Habbu, Narayan Miskin1, Venkatrao H. Kulkarni, Pradeep Bhat, Arun Joshi, Anant Bhandarkar, Satish Kulkarni, Sheshagiri R. Dixit, Jaishree Vaijanathappa

DOI: 10.7324/JAPS.2020.103018Pages: 135-148

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In silico and in vitro assay of Hexagamavunon-6 analogs, Dibenzilyden-N-Methyl-4-piperidone as antibacterial agents

Tesia Aisyah Rahmania, Ritmaleni Ritmaleni, Erna Prawita Setyowati

DOI: 10.7324/JAPS.2020.103004Pages: 039-043

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Growth inhibition of combined treatment of cationic liposome/p53 complexes and cisplatin on human carcinoma cells

Wanlop Weecharangsan, Robert J. Lee

DOI: 10.7324/JAPS.2020.104006Pages: 034-040

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Fenugreek (Trigonella foenum-graceum) increases postmenopausal fibroblast-associated COL1A1 and COL3A1 production dominantly through its binding to estrogen receptor beta

Shannaz Nadia Yusharyahya, Kusmarinah Bramono, Andon Hestiantoro, Sarah Qanita Edwar, Indra Kusuma

DOI: 10.7324/JAPS.2020.104004Pages: 022-027

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Identification, synthesis, and characterization of β-isomer as process related impurity in production of methocarbamol from guaifenesin

Appala Raju Nemala, Sridevi Chigurupati, Kesavanarayanan Krishnan Selvarajan, Saurabh Bhatia, Sridevi Pingali, Anitha Sadula

DOI: 10.7324/JAPS.2020.10502Pages: 010-015

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3D QSAR and docking studies on benzoylsulfonohydrazides as histone acetyltransferase KAT6A inhibitors

MD. Muzaffar-Ur-Rehman, Syed Akbar, Asra Ali Bahazeq

DOI: 10.7324/JAPS.2020.10504Pages: 023-030

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Novel aminoalkylated chalcone: Synthesis, biological evaluation, and docking simulation as potent antimalarial agents

Jufrizal Syahri, Hasmalina Nasution, Beta Achromi Nurohmah, Bambang Purwono, Emmy Yuanita

DOI: 10.7324/JAPS.2020.10601Pages: 001-005

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Synthesis and biological evaluation of novel substituted pyrrolo[2,3-d]pyrimidines as anticancer agents

Sandip P. Dholakia, Kaushik B. Kanada, Ghanshyam R. Parmar

DOI: 10.7324/JAPS.2020.10602Pages: 006-011

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Effect of illness perception on improving asthma symptoms with omega-3 fish oil therapy: Pre-post design

Amelia Lorensia, Mariana Wahyudi, Ananta Yudiarso, Siti Erfina Dwi Kurnia

DOI: 10.7324/JAPS.2020.10609Pages: 062-071

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Lapatinib-loaded nanocolloidal polymeric micelles for the efficient treatment of breast cancer

Gunjan Vasant Bonde, Gufran Ajmal, Sarita Kumari Yadav, Pooja Mittal, Brahmeshwar Mishra

DOI: 10.7324/JAPS.2020.10903Pages: 023-029

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Insights into the structural features of anticancer 1,6-naphthyridines and pyridopyrimidines as VEGFR-2 inhibitors: 3D-QSAR study

Siddharth J. Modi, Dharti H. Modh, Vithal M. Kulkarni

DOI: 10.7324/JAPS.2020.10101Pages: 001-022

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Approaches for synthesis and chemical modification of non-condensed heterocyclic systems based on 1,3,4-oxadiazole ring and their biological activity: A review

Maryan Lelyukh, Marta Martynets, Myroslava Kalytovska, Iryna Drapak, Stefan Harkov, Taras Chaban, Ihor Chaban, Vasyl Matiychuk

DOI: 10.7324/JAPS.2020.1010016Pages: 151-165

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In silico studies on pyrazine derivatives for identifying potential inhibitors of PIM-1 kinase

Amena Ali, Abuzer Ali, Mohd. Washid Khan, Abutahir, Ibraheem Husain, Kuldeep Patel, Vivek Asati

DOI: 10.7324/JAPS.2020.10116Pages: 040-049

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Study of alterations in pharmacokinetics and pharmacodynamics of Saxagliptin in the presence of Rutin: An interaction study in rats

Naga Raju Kandukoori, Pavani Uppu, Narsimha Reddy Yellu

DOI: 10.7324/JAPS.2020.101111Pages: 081-086

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Synthesis and cytotoxic evaluation of novel chromenes and chromene(2,3-d)pyrimidines

Mahmoud N. M. Yousif, Abdel-Rahman B. A. El-Gazzar, Ahmed A. Fayed, May A. El-Manawaty, Nabil M. Yousif

DOI: 10.7324/JAPS.2020.101205Pages: 035-043

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Bioguided study of the Antarctic alga Himantothallus grandifolius (A. Geep & E.S.Geep) indicates 13E-Docosenamide as potential antileishmanial agent

Leandro Costa Clementino, Fabio Aurelio Esteves Torres, Angela Maria Arenas Velasquez, Leonardo Villela, Toyota Fujii Mutue, Pio Colepicolo, Marcia A. S. Graminha

DOI: 10.7324/JAPS.2020.101213Pages: 098-103

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New benzothiazinone linked 1, 2, 4-triazoles: Design, synthesis, characterization, and evaluation of antitubercular activity

Kannampally Ajmal, Gurubasavaraj V. Pujar, Sethu Arun Kumar, Subhankar P. Mandal, Manisha Singh

DOI: 10.7324/JAPS.2021.110204Pages: 029-038

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Cytotoxicity of Quercetin and Quercetin-3-O-rhamnoside of Etlingera elatior (Jack) R.M.Sm. leaves against HeLa Cervical Cancer Cells

Herni Kusriani, Anas Subarnas, Ajeng Diantini, Yoppi Iskandar

DOI: 10.7324/JAPS.2021.110512Pages: 085-090

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WRL-68 with the overexpression of CYP3A4 as an in vitro model to assess drug–drug interaction

Nurliana Abd Mutalib, Normala Abd Latip

DOI: 10.7324/JAPS.2021.110408Pages: 057-067

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Antibacterial evaluation and molecular properties of pyrazolo[3,4-b] pyridines and thieno[2,3-b]pyridines

Mervat A. Elsherif

DOI: 10.7324/JAPS.2021.110614Pages: 118-124

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Growth inhibition of cholic acid-conjugated polyethylenimine 25K/ p53-EGFP complexes on human carcinoma cells

Wanlop Weecharangsan, Nattisa Niyomtham, Boon-ek Yingyongnarongkul, Praneet Opanasopit, Robert J. Lee

DOI: 10.7324/JAPS.2021.110403Pages: 014-021

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Micropatterned κ-carrageenan-PVP-PEG hydrogels as a templet for head and neck cancer spheroid culture

Nadia Halib, Zainah Adam, Maznah Mahmud

DOI: 10.7324/JAPS.2021.110503Pages: 015-021

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Nephroprotectivity of Coccinia indica leaves against gentamycin-induced nephrotoxicity using in vitro and in vivo models

Neelima Satrasala, Dwarakanadha Reddy Peram, Chandra Sekhar Kothapalli Bannoth

DOI: 10.7324/JAPS.2021.110616Pages: 132-139

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Isolation, peroxisome proliferator-activated receptor-gamma transcription, glucose uptake, and molecular docking of tetramethoxyflavonoids from the leaves of Rourea mimosoides (Vahl) Planch.

Che Puteh Osman, Norhafizoh Abdul Somat, Zuriati Zahari, Syahrul Imran, Mohd Ilham Adenan

DOI: 10.7324/JAPS.2021.110802Pages: 010-016

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Immunopotentiation of galangal (Alpinia galanga L.) when combined with T-cells against metastatic triple-negative breast cancer, MDA-MB 231

Iffan Alif, Rohmad Yudi Utomo, Faradiba Nur Ahlina, Nadzifa Nugraheni, Dedy Hermansyah, Agung Putra, Edy Meiyanto

DOI: 10.7324/JAPS.2021.1101107Pages: 053–061

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Design, synthesis and in silico prediction of drug-likeness properties of new ortho, meta and para-(2-cyano-3-(3,5-di-tert-butyl-4- hydroxyphenyl)acrylamido)benzoic acids

Madhavi Kuchana, Lakshmi Bhavani Kambala

DOI: 10.7324/JAPS.2021.110805Pages: 031-035

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Novel glitazone attenuates rotenone-induced toxicity in mouse model of Parkinson’s disease

Ankith B. Shetty, Kamsagara Linganna Krishna, Bommenahally Ravanappa Prashantha Kumar, Hittanahalli Shivakumar Nandini

DOI: 10.7324/JAPS.2021.1101007Pages: 042-049

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Prevalence of OCT1 (rs628031) genetic polymorphism in south Indian population

Swathi Swaroopa Borra, Bhavya Chebrolu, Poojitha Thotakura, Sujin Bright Francis Joice, Vasanth Raj Palanimuthu, Sadagoban Gopal Krishnamoorthy, Arun Kanniyappan Parthasarathy

DOI: 10.7324/JAPS.2021.1101006Pages: 035-041

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Nanodelivery systems for Alzheimer's disease: Prospects of natural therapeutic agents

Oluwatoyin A. Odeku, Tolulope O. Ajala

DOI: 10.7324/JAPS.2021.1101101Pages: 001-010

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Biochemical characterization and ecofriendly field application of the plant growth-promoting rhizobacterium Bacillus amyloliquefaciens MH046937 isolated from Salsola imbricata in Tur Sinai, Egypt

Warda E. Ashour, Moustafa M. Zohair, Ahmed A. El-Beih, Eman R. Hamed, Abeer A. Abd El Aty

DOI: 10.7324/JAPS.2021.120109Pages: 094-105

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Analysis of the literature on 3D printing in healthcare with reference to pharmaceuticals using a bibliometric approach

Virendra S. Ligade, Akash Chimegave

DOI: 10.7324/JAPS.2022.120310Pages: 096–102

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Preparation and evaluation of novel self-dispersing lipid formulation of nevirapine for oral delivery

Gopalapura Bellaiah Preethi, Hagalavadi Nanjappa Shivakumar, Madalli Ravi Kumar

DOI: 10.7324/JAPS.2022.120313Pages: 123–131

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The glucose uptake of type 2 diabetic rats by Sargassum olygocystum extract: In silico and in vivo studies

Muhamad Firdaus, Rahmi Nurdiani , Bachtiar Rivai, Windy Hapsari Hemassonida, Aqilatul Badzliyah, Nur Khasanah Sugiat

DOI: 10.7324/JAPS.2022.120314Pages: 132–139

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Phytochemical screening, docking study, and in vitro assessment of cytotoxicity against MCF7 and 3T3 cell lines of Indonesian sea cucumber Stichopus sp.

Teni Ernawati , Minarti Minarti, Galuh Widiyarti, Megawati Megawati, Faiza Maryani

DOI: 10.7324/JAPS.2022.120411Pages: 096-107

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Overexpression of soluble recombinant Thermus thermophilus (Tth) DNA polymerase in Escherichia coli BL21(DE3) using an MBP fusion tag as a solubility enhancer

Iman Permana Maksum, Diandra Firdiani Utami, Eva Annisa Nurhakim, Yosua, Sriwidodo, Muhammad Yusuf, Muhammad Fadhlillah, Ryan Adibagus Haryanto

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In vitro antiplasmodial activities of the fractions of Hyrtios reticulatus sponge extract

Mahfur Mahfur, Indah Purwantini, Subagus Wahyuono, Erna Prawita Setyowati

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Impact of Morus alba L. on the expression of drug-metabolizing enzymes and transporters in Caco-2 cells

Waranya Chatuphonprasert, Wipawee Tukum-mee, Jintanaporn Wattanathorn, Kanokwan Jarukamjorn

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