Review on Biological Activities of 1,3,4-Thiadiazole Derivatives
Arvind k. Singh, Geeta Mishra, Kshitiz Jyoti
Pages: 44-49
Epigenetic modification of suppressor of cytokine signaling-3 in asthmatic mouse lung: role of interleukin-6
Vani Mishra, Rahul Sharma, Brajadulal Chattopadhyay, Bhola Nath Paul
Pages: 81-89
Synthesis and in-vitro screening of 3,4-dihydropyrimidin-2(1H)-one derivatives for antihypertensive and calcium channel blocking activity
Hiren M. Marvaniya, Palak K. Parikh, Dhrubo Jyoti Sen
Pages: 109-113
Synthesis, characterization and anti-trypanosomal activity of R-(-)carvone and arylketones-thiosemi carbazones and toxicity against Artemia salina Leach
Bienvenu Glinma, Salome D. S. Kpoviessi, Raymond H. Fatondji, Fernand A. Gbaguidi, Coco N. Kapanda, Joanne Bero, Didier M. Lambert, Veronique Hannaert, Joëlle Quetin-Leclercq, Mansourou Moudachirou, Jacques Poupaert, Georges C. Accrombessi
Pages: 65-70
Enhancement of camptothecin production in Camptotheca acuminata hairy roots by overexpressing ORCA3 gene
Xiaoning Ni, Shiqiu Wen, Wei Wang, Xiaoyun Wang, Hui Xu, Guoyin Kai
Pages: 85-88
Antifungal activity of bioactive compound of seeds of Psoralea corylifolia L. against seed borne Fusarium species of maize
Kiran. B, Lalitha.V, Raveesha.K.A
Pages: 161-164
Histological Studies in Murine Model of Asthma: Effect of Stat3 siRNA
Bhushan Chaudhari, Pankaj Jagdale, Sheikh Raisuddin, Shambhoo Sharan Tripathi, Mamta Shukla, Pradeep Kumar Singh, Pradeep Kumar
Pages: 77-84
Gastro-Retentive Floating Matrix Tablets of Cefpodoxime Proxetil
K. Sreenivasa Rao, Rakesh R. Vairagkar, Dattatreya B. Udgirkar, Praveen S. Patil, Karnakumar V. Biradar
Pages: 190-194
Improving Oral Bioavailability of Agaricoglycerides by Solid Lipid-Based Self-Emulsifying Drug Delivery System
Chun Chao Han, Linna Han
Pages: 195-199
Antihyperlipidaemic Activity of Spermacoce Hispida Ethanolic Extract in Triton WR-1339 Induced Hyperlipidaemic Rats
G. Sivaelango, P. Senthil Kumaran, P. Kumaravel, P. Revathi, A. Jaswant
Pages: 95-98
Genotoxicity of anticancer drug Azathioprine (Imuran): role of Omega-3 (?-3) oil as protective agent
Elelaimy I.A, Elfiky S.A., Hassan A.M., Ibrahim H.M., Elsayad R.I.
DOI: 10.7324/JAPS.2012.2404Pages: 14-23
Community Pharmacy/Hospital Based Assessment of Clinical Pharmacist Intervention for Safe and Effective Drug Use
Awofisayo Sunday Olajide, Aboyarin Oladayo, Udoh Imo Emmanuel
DOI: 10.7324/JAPS.2012.2424Pages: 66-69
GC-MS analysis of Polygala rosmarinifolia Wights & Arn
M. Alagammal, P. Tresina Soris, V.R. Mohan
DOI: 10.7324/JAPS.2012.2504Pages: 188-190
In-Vitro Anthelmintic Activity of Croton Bonplandianum Baill
Hapse S.A., Pagar H.J. Suruse S.D., Ugale S.S.
DOI: 10.7324/JAPS.2012.2516Pages: 191-193
Comparative in vitro antibacterial activities study of some mucoadhesive polymeric suspensions containing fluoroquinolones
Chandra Kanti Chakraborti, Subhashree Sahoo, Pradipta Kumar Behera, Anjulata Manjari Sahoo
DOI: 10.7324/JAPS.2012.2502Pages: 44-48
Simultaneous determination of pioglitazone and glimepiride in their pharmaceutical formulations
Mamdouh R. Rezk, Safa'a M. Riad, Ghada Y. Mahmoud, Abdel-Aziz El Bayoumi Abdel Aleem
DOI: 10.7324/JAPS.2012.2544Pages: 177-184
Synthesis and antimicrobial activity of novel (3,5-dichloro-4-((5-aryl-1,3,4-thiadiazol-2-yl)methoxy) phenyl) aryl methanones
V. Srinivasa Murthy, B. K. Manuprasad, S. Shashikanth
DOI: 10.7324/JAPS.2012.2726Pages: 172-176
Chemical Constituents of the Essential Oil of Laggera pterodonta (DC.) Sch. Bip. From North-Central Nigeria
Egharevba Henry Omoregie, Kunle Folashade Oluyemisi, Okwute Simon Koma, Okogun Joseph Ibumeh
DOI: 10.7324/JAPS.2012.2835Pages: 198-202
Isolation of a novel triterpene from the Essential oil of fresh leaves of Chromolaena odorata and its in-vitro cytotoxic activity against HepG2 cancer cell line
Velliangiri Prabhu and Subban Ravi
DOI: 10.7324/JAPS.2012.2926Pages: 132-136
Synthesis of novel Naphthalene COX inhibitors for anti-inflammatory activity
Anand B. Pandya, Dhaval G. Prajapati, Saurabh S. Pandya
DOI: 10.7324/JAPS.2012.2840Pages: 226-232
HPLC evaluation on 3-n-butylphthalide distribution
Qi Wang, Shuoyang Li, Peifeng Liu, Ming Shen, Tao Gong, Yourong Duan, Zhang Zhi-Rong
DOI: 10.7324/JAPS.2012.21003Pages: 016-020
Anti-ischemic effect of ethyl acetate extract of Aquilaria crassna by attenuation of p38-MAPK activation
Chanyatip Suwannasing, Nitchawat Paiyabhroma, Sarawut Kumphune
DOI: 10.7324/JAPS.2012.21005Pages: 026-030
Three component one pot synthesis of 5-Substituted 1-Aryl-2,3-diphenyl imidazoles: A novel class of promising antioxidants
Nagaraja Naik, H. Vijay Kumar, J. Rangaswamy, S.T. Harinia and T.C. Umeshkumar
DOI: 10.7324/JAPS.2012.21112Pages: 067-074
3',4'-Dimethoxy Quercetin, a Flavonol Compound Isolated from Kalanchoe pinnata
Akhmad Darmawan, Megawati and Sofa Fajriah
DOI: 10.7324/JAPS.2013.30116Pages: 088-090
Synthesis and Antihypertensive Activity of Some Quinazoline Derivatives
Harsha U. Patel, Ravi S. Patel, Chhaganbhai N. Patel
DOI: 10.7324/JAPS. 2013.30332Pages: 171-174
Study of Complex Nutrients, Temperature and Salts on Hyaluronic acid Production In Streptococcus zooepidermicus ATCC 43079
Nguyen Tu Hoang Khue and Pham Thien Minh Vo
DOI: 10.7324/JAPS.2013.3503Pages: 012-015
Formulation and In-Vitro Characterization of Acyclovir Floating Matrix Tablets: A Factorial Design Study
Sadhana Shahi, Ashok Sonawane, Suhas Vanamore, Nityanand Zadbuke
DOI: 10.7324/JAPS.2013.3513Pages: 065-074
Possible Involvement of 'Phosphatidylinositol-3 kinase and endothelial nitric oxide synthase' in experimental obesity induced vascular endothelium dysfunction
Gargee Dubey, PL Sharma and Saurabh Sharma
DOI: 10.7324/JAPS.2013.3608Pages: 052-060
Glypican-3 as a tumor marker for hepatocellular carcinoma
Amal A. Mohamed, Naglaa El-Toukhy, M. Magdi Atta, Salah M. Ahmed
DOI: 10.7324/JAPS.2013.3613Pages: 083-087
Exopolysaccharide in Lactobacillus Rhamnosus Pn04 After Co-Culture with Leuconostoc mesenteroides Vtcc-B-643
Nguyen Tu Hoang Khue and Nguyen Huu Ngoc
DOI: 10.7324/JAPS.2013.3703Pages: 014-017
Measuring Interesting Amino Acid Patterns for Alzheimer's Disease Related Studies Targets on the Binding Site Using Association Rule Mining
D. Ponmary Pushpa Latha and D. Joseph Pushpa Raj
DOI: 10.7324/JAPS.2013.3705Pages: 025-030
Determination of Total Arsenic in Indonesian Tuna Fish Sample
Tiny A. Koesmawati, B. Buchari, Muhammad B. Amran, Leonardus B.S. Kardono
DOI: 10.7324/JAPS.2013.3722Pages: 116-121
Microwave assisted synthesis of 3-α-carboxy ethylrhodanine derivatives and their in vitro antibacterial activity
Kaveri Sundaram and Subban Ravi
DOI: 10.7324/JAPS.2013.3725Pages: 133-135
Enteric coating of hard gelatin capsules by the spouted bed process
H.V.A. Oliveira, M.P.G. Peixoto, L.A. Tacon & L.A.P.Freitas
DOI: 10.7324/JAPS.2013.3810Pages: 057-063
Statistical Optimization of Olanzapine Ternary Solid Dispersions with Pvp K 30 and Peg 20,000 by Response Surface Methodology
Anil Katharia, Ratendra Kumar, Rajiv Sharma, Yogendra Singh, Uday Veer Singh Teotia
DOI: 10.7324/JAPS.2013.3920Pages: 109-116
In silico Analysis of 3D-QSAR and Molecular Docking for Bcl-2 Inhibitors to Potential Anticancer Drug Development
Ramachandran M, Balwin Nambikkairaj, Kumaran K, Arun Kumar De and G.Ramesh Kumar
DOI: 10.7324/JAPS.2013.31005Pages: 023-029
Efficacy of 5-(2-aroyl)aryloxy methyl-2-phenyl-1,3,4-oxadiazoles as antibacterial and antifungal agents
Bushra Begum A, Noor Fatima Khanum, Naveen P, Lakshmi Ranganatha V, Asha MS and Shaukath Ara Khanum
DOI: 10.7324/JAPS.2013.31119Pages: 105-109
Cytotoxic effects of antiglypican-3 against HepG2 cell line
Randa A Zaghloul, Mohammed M H Al-Gayyar, Mamdouh M El-Shishtawy, Mohamed A. Ebrahim
DOI: 10.7324/JAPS.2013.31206Pages: 031-035
3D QSAR and Pharmacophore Modelling on Chalcones as Antileishmanial Agents potential Trypanothione reductase Inhibitors
Sujit Arun Desai, Santosh Sahedeo Kumbhar, Vishal Shankar Katti, Prafulla Balkrishna Choudhari, Manish Sudesh Bhatia
DOI: 10.7324/JAPS.2013.31218Pages: 099-102
Computational analysis of phytocompounds with 1,3-β-D-Glucan synthase for antidermatophytic activity
M Jeyam, M Arangaraj, P Ravikumar, G Shalini
DOI: 10.7324/JAPS.2014.40211Pages: 064-069
Synthesis of Methyl 2-Cinnamamido-3-Hydroxy Propanoate Having Activity against P388 Leukemia Cells
Teni Ernawati, Yulia Anita, Puspa Dewi Lotulung and Muhammad Hanafi
DOI: 10.7324/JAPS.2014.40318Pages: 092-095
Effect of formulation parameters on Sumatriptan succinate Buccal Mucoadhesive Tablet: Quality by Design approach
Wable Arti J, Thokal Seema B, Mittal Sandeep S, Shirsat Ajinath E, Bhingare Chandrashekhar L, Ingle Pramod L
DOI: 10.7324/JAPS.2014.40418Pages: 103-111
In vitro cytotoxicity effects of single and combination Nigella sativa and Zingiber zerumbet extracts on human myeloid leukemia (HL60) cells and its mode of cell death
Norfazlina M.N., Farida Zuraina M.Y., Rajab N.F, Mohd Nazip S., Rumiza A.R., Suziana Zaila C.F., Lek Mun L., Nurshahirah N., Florinsiah L.
DOI: 10.7324/JAPS.2014.40509Pages: 051-055
Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines
Guillaume Burgy, Emmanuelle Limanton, François Carreaux, Emilie Durieu, Laurent Meijer, and Jean-Pierre Bazureau
DOI: 10.7324/JAPS.2014.40604Pages: 025-032
Cytotoxic activity and apoptosis induction of 8-hydroxyisocapnolactone-2´,3´-diol and its combination with Doxorubicin on MCF-7 and T47D cells
Ratna Asmah Susidarti, Riris Istighfari Jenie, Muthi’ Ikawati, Dyaningtyas Dewi Pamungkas Putri, Edy Meiyanto
DOI: 10.7324/JAPS.2014.40614Pages: 089-097
Piceatanol: Anti-Cancer Compound From Gewang Seed Extract
Leny Heliawati, Agus Kardinan, Tri Mayanti, Roekmi-ati Tjokronegoro
DOI: 10.7324/JAPS.2015.50119Pages: 110-113
Evaluation as antioxidant agents of 1,2,4-triazole derivatives: effects of essential functional groups
Ahmet Cetin, Ibrahim Halil Geçibesler
DOI: 10.7324/JAPS.2015.50620Pages: 120-126
Formulation and in vitro evaluation of berberine containing liposome optimized by 32 full factorial designs
Girish Sailor, A K Seth, Ghanshyam Parmar, Sachin Chauhan, Ankur Javia
DOI: 10.7324/JAPS.2015.50704Pages: 023-028
Chemical Constituents of Cordia dichotoma G. Forst.
Consolacion Y. Ragasa, Virgilio Ebajo Jr., Mariquit M. De Los Reyes, Emelina H. Mandia, Maria Carmen S. Tan, Robert BrkljaÄa, Sylvia Urban
DOI: 10.7324/JAPS.2015.58.S3Pages: 016-021
Chemical constituents of Cycas aenigma
Vincent Antonio S. Ng, Esperanza Maribel G. Agoo, Chien-Chang Shen, Consolacion Y. Ragasa
DOI: 10.7324/JAPS.2015.50906Pages: 032-036
Synthesis and screening of new maleimide derivatives as potential anti-tubercular agents
Saroj Kumar Sahoo, Kurre Purna Nagasree, Jamullamudi Risy Namratha, Pemmadi Raghuveer Varma, Muthyala Murali Krishna Kumar
DOI: 10.7324/JAPS.2015.510.S8Pages: 044-047
In silico analysis of indole-3-carbinol and its metabolite DIM as EGFR tyrosine kinase inhibitors in platinum resistant ovarian cancer vis a vis ADME/T property analysis
Raju Dash, S. M. Zahid Hosen, Md. Rezaul Karim, Mohammad Shah Hafez Kabir, Mohammed Munawar Hossain, Md. Junaid, Ashekul Islam, Arkajyoti Paul, Mohammad Arfad Khan
DOI: 10.7324/JAPS.2015.501112Pages: 073-078
Pharmacokinetics interaction of dapoxetine with different doses of green tea extract in male healthy volunteers using midazolam as CYP3A4 enzyme probe
Khaled Sobhy Abdelkawy, Ahmed M Donia, Mahmoud S Abdallah
DOI: 10.7324/JAPS.2015.501201Pages: 001-007
Cytotoxic effect and apoptotic activity of Parmentiera edulis DC. hexane extract on the breast cancer cell line MDA-MB-231
Cynthia Carolina Estanislao Gómez, Cynthia Ordaz Pichardo, Eduardo San Martín Martínez, Nury Pérez Hernández, Guillermo Pérez Ishiwara, María del Consuelo Gómez García
DOI: 10.7324/JAPS.2016.600103Pages: 015-022
Synthesis, Evaluation and Docking Study of 1, 3, 5-Triazine Derivatives as Cytotoxic Agents against Lung Cancer
Marwa F. Balaha, Mervat H. El-Hamamsy, Nabawya A. Sharaf El-Din, Nageh A.El-Mahdy
DOI: 10.7324/JAPS.2016.60405Pages: 028-045
Synthesis and antibacterial activity of novel 2-(arylimino)thiazolidin-4-one and 2-(benzylidenehydrazono)-3-arylthiazolidin-4-one derivatives
Ebaa M. El-Hossary, Yassin M. Nissan, Katharina Edkins, Heike Bruhn
DOI: 10.7324/JAPS.2016.60502Pages: 007-017
Production of antioxidant xylooligosaccharides from lignocellulosic materials using Bacillus amyloliquifaciens NRRL B-14393 xylanase
Mona M. Rashad, Abeer E. Mahmoud, Mohamed U. Nooman, Hadeer A. Mahmoud, Alaa El-Din M.M. El-Torky, Akaber T. Keshta
DOI: 10.7324/JAPS.2016.60606Pages: 030-036
A preliminary evaluation of anticancer and antioxidant potential of two traditional medicinal plants from Lamiaceae-Pogostemon heyneanus and Plectranthus amboinicus
Vaishali Rai, Vinitha Ramanath Pai, Pratapchandra Kedilaya
DOI: 10.7324/JAPS.2016.60811Pages: 073-078
Mechanism of Relaxant Action of Ethyl 6-amino-5-cyano-2-methyl- 4-(pyridin-4-yl)-4H-pyran-3-carboxylate Mainly Through Calcium Channel Blockade in Isolated Rat Trachea
Soledad Alemán-Pantitlán, César Millán-Pacheco, Miguel A. Vázquez, Fernando Hernández-Borja, Rafael Villalobos-Molina, Blanca Bazán-Perkins, Samuel Estrada-Soto
DOI: 10.7324/JAPS.2016.601004Pages: 029-036
Synthesis, spectroscopic characterization and biological applications of Cu(II) and Ni(II) complexes with 2-butyl-4-chloro-5-formylimidazole thiosemicarbazone
A. Sreenath Reddy, L. Sivarama Krishna, H. K. Rashmi, P. Uma Maheswari Devi, Y. Sarala, A. Varada Reddy
DOI: 10.7324/JAPS.2016.601015Pages: 107-112
Clonazepam associated hypothyroidism: Aforethought on a concealed dilemma
Rupam Gill, Dipanjan Bhattacharjee, Navin A. Patil, Shripathy M. Bhat
DOI: 10.7324/JAPS.2016.601031Pages: 222-225
Antifeedant Constituents from Leucaena leucocephala
Poonam Negi, Bhupendra Singh Rawat, Devendra Singh Negi
DOI: 10.7324/JAPS.2016.601204Pages: 028-031
Effect of intensive endurance training on rat brain and hepatic 8-oxoguanine DNA glycosylase and 8-hydroxy-2'-deoxyguanosine levels
Mohammad Esmaiel Afzalpour, Hossein TaheriChadorneshin, Seyed-Hosein Abtahi-Eivary, Ehsan Afroozi-Gerow
DOI: 10.7324/JAPS.2016.601215Pages: 110-113
Nanochemopreventive effect of polymer functionalized gold nanoparticles containing hesperetin drug inhibited proliferation and induced apoptosis in Hep3B cells
Gokuladhas Krishnan, Jayakumar Subramaniyan, Pramila Chengalvarayan Subramani, Devaki Thiruvengadam
DOI: 10.7324/JAPS.2016.601216Pages: 114-123
Effect of exogenous application of indole-3-acetic acid (IAA) on cell maturity of Olea europaea L. and extractability of phenolic compounds in virgin olive oil
Youssef MOUSTAKIME, Zakaria HAZZOUMI, Zain El Abidine FATEMI, Khalid AMRANI JOUTEI
DOI: 10.7324/JAPS.2017.70228Pages: 199-206
QSAR and Molecular Docking of Phthalazine Derivatives as Epidermal Growth Factor Receptor (EGFR) Inhibitors
Monika G. Shinde, Siddharth J. Modi, Vithal M. Kulkarni
DOI: 10.7324/JAPS.2017.70427Pages: 181-191
Synthesis and evaluation of silver nanoparticles using Cymodocea rotundata against clinical pathogens and human osteosarcoma cell line
Jayanthi Abraham, Shantanu Saraf, Vakas Mustafa, Yugal Chaudhary, Silambarasan Sivanangam
DOI: 10.7324/JAPS.2017.70608Pages: 055-061
Synthesis and antimicrobial activity of Bis-Derivatives of 3a′, 6a′Dihydro-2'H-Spiro[Indole-3,1'-Pyrrolo[3,4-c]Pyrrole]-2,4',6'(1H, 3'H, 5'H)-Trione
Ruslan Gr. Redkin, Evgeniya I. Syumka, Leonid A. Shemchuk, Valentin P. Chernykh
DOI: 10.7324/JAPS.2017.70610Pages: 069-078
Design, Synthesis and Preliminary Pharmacological Screening (antimicrobial, analgesic and anti-inflammatory activity) of Some Novel Quinazoline Derivatives
Biswajit Dash, Suvakanta Dash, Damiki Laloo, Chitrani Medhi
DOI: 10.7324/JAPS.2017.70612Pages: 083-096
Evaluation of Plant Food Extracts in Experimental Model of Alzheimer's Like Disease Induced by Aluminum Lactate in Rats
Sahar Y. Al-Okbi, Doha A. Mohamed, Mohamed Abdel Fatah, Kholoud Abdel Aal, Shaimaa E Mohammed
DOI: 10.7324/JAPS.2017.70712Pages: 070-076
Computational, structural and functional aspects of hypothetical protein of Aspergillus flavus Pheromone Receptor Pre-A (PRP-A)
Maneesh Kumar, Sindhuprava Rana, Harish Kumar, Pratik Kumar, Manas Ranjan Dikhit, Rani Mansuri, Jainendra Kumar, Ganesh Chandra Sahoo
DOI: 10.7324/JAPS.2017.70714Pages: 089-097
Synthesis and establishment of Amlodipine impurity G reference standard
Ly Dieu Ha, Trang Thi Diem Nguyen, Tri Minh Le
DOI: 10.7324/JAPS.2017.71015Pages: 105-110
Anticancer Activity of New Substituted Pyrimidines, Their Thioglycosides and Thiazolopyrimidine Derivatives
Mahmoud N. M. Yousif, Wael A. El-Sayed, Hebat-Allah S. Abbas, Hanem M. Awad, Nabil M. Yousif
DOI: 10.7324/JAPS.2017.71104Pages: 021-032
Steroids and isoquercetin from Lygodium microphyllum
Hadi Kuncoro, Kindi Farabi, Laode Rijai
DOI: 10.7324/JAPS.2017.71120Pages: 136-141
QSAR, Molecular Docking and Dynamics Studies of Pyrrolo[2,3-b]Pyridine Derivatives as Bruton’s Tyrosine Kinase Inhibitors
Ruslin, Nirwana, Muhammad Arba, Mukhsar, Daryono Hadi Tjahjono
DOI: 10.7324/JAPS.2017.71201Pages: 001-007
Accessing the Anti-Proliferating Activity of Tankyrase-2 Inhibitors via 2D, 3D-QSAR and Molecular Docking: Assessment of Structure Activity Relationships
Mervat H. El-Hamamsy
DOI: 10.7324/JAPS.2017.71203Pages: 014-027
Quality of Life Assessment in Cancer Patients of Regional Centre of Hyderabad City
V. Naga Sunanda M. Priyanka, J. Architha1 , M. Shravan, A. Srinivasa Rao, Mohd. Abdul Hadi
DOI: 10.7324/JAPS.2018.8125Pages: 165-169
Anti-inflammatory and antioxidant activity of salicylic acid conjugated dihydropyrazoline analogues
Naveen Puttaswamy, Rekha N D, Lakshmi Ranganatha V, Prashanth T, Shaukath Ara Khanum
DOI: 10.7324/JAPS.2018.8209Pages: 060-064
Alkaline Phosphatase Activity of Marsilea crenata Presl. Extract and Fractions as Marker of MC3T3-E1 Osteoblast Cell Differentiation
Burhan Ma’arif, Mangestuti Agil, Hening Laswati
DOI: 10.7324/JAPS.2018.8308Pages: 55-59
Computational Model of Doxorubicin Conjugate with Docosahexaenoic Acid and Integrin αvβ3 Ligand for Anticancer
Ace T. Hidayat, Muhammad Yusuf, Husein H. Bachti, Ajeng Diantini, Achmad Zainuddin
DOI: 10.7324/JAPS.2018.8401Pages: 001-006
Cisplatin-Induced Nephrotoxicity in Rats: Modulatory Role of Simvastatin and Rosuvastatin against Apoptosis and Inflammation
Rasha E. Mostafa, Dalia O. Saleh, Dina F. Mansour
DOI: 10.7324/JAPS.2018.8406Pages: 043-050
Molecular Docking Studies Involving the Inhibitory Effect of Gymnemic Acid, Trigonelline and Ferulic Acid, the Phytochemicals with Antidiabetic Properties, on Glycogen Synthase Kinase 3 (α and β)
V. Roshana Devi, C. Sharmila, S. Subramanian
DOI: 10.7324/JAPS.2018.8422Pages: 150-160
QSAR, Molecular Docking and Dynamics Studies of Quinazoline Derivatives as Inhibitor of Phosphatidylinositol 3-Kinase
Muhammad Arba, Ruslin, Waode Umi Kalsum, Armid Alroem, Muhammad Zakir Muzakkar, Ida Usman, Daryono Hadi Tjahjono
DOI: 10.7324/JAPS.2018.8501Pages: 001-009
Synthesis and Evaluation of Antimitotic Activity of N-Phenyl Tetralones
Umesha Basavaiah, Sowbhagya, Vinaya, Yeriyur Basavaiah Basavaraju
DOI: 10.7324/JAPS.2018.8512Pages: 094-100
Design, One-pot Synthesis and Biological Evaluation of Imidazo[2,1-b] [1,3,4] Thiadiazole Derivatives for their Anti- Tubercular and Anti-Fungal Activity
Manjoor Ahamad Syed, Yiragam Reddy Padmanabha Reddy, K. B. Chandrasekhar
DOI: 10.7324/JAPS.2018.8704Pages: 021-027
Effect of Kirganelia reticulata extract on Human Embryonic Kidney cells with evidence on morphological changes
Madhurima Ghosh, Jhinuk Chatterjee, V. Krishnamurthy
DOI: 10.7324/JAPS.2018.8917Pages: 114-118
3D-QSAR analysis of pyrimidine derivatives as AXL kinase inhibitors as anticancer agents
Siddharth J. Modi, Vithal M. Kulkarni
DOI: 10.7324/JAPS.2018.81103Pages: 015-027
Effects of sea urchin (Diadema setosum) gonad extracts on gene expression of FOXP3 and the production of cytokine on Salmonella typhi-induced mice
Wa Ode Salma, Sitti Wahyuni, Nursin Kadir, Suryani Asad, Irawan Yusuf 
DOI: 10.7324/JAPS.2018.81216Pages: 140-146
In silico evaluation of Benzo (f) chromen-3-one as a potential inhibitor of NF-κB: A key regulatory molecule in inflammation-mediated pathogenesis of diabetes, Alzheimer’s, and cancer
Sandeep Kumar Gandham, Venkata Ramaiah Chintha, Rajendra Wudayagiri
DOI: 10.7324/JAPS.2018.81218Pages: 157-164
3D-QSAR, molecular docking, and dynamics simulation of quinazoline–phosphoramidate mustard conjugates as EGFR inhibitor
Ruslin Ruslin, Resky Amelia, Yamin Yamin, Sandra Megantara, Chun Wu, Muhammad Arba
DOI: 10.7324/JAPS.2019.90113Pages: 089-097
In silico predictive for modification of chalcone with pyrazole derivatives as a novel therapeutic compound for targeted breast cancer treatment
Riska Prasetiawati, Adel Zamri, Melisa Intan Barliana, Muchtaridi Muchtaridi
DOI: 10.7324/JAPS.2019.90203Pages: 020-028
Qualitative anti-tubercular activity of synthetic ethyl 7-acetyl2-substituted-3-(4-substituted benzoyl) indolizine-1-carboxylate analogues
Sandeep Chandrashekharappa, Katharigatta N. Venugopala, Rashmi Venugopala, Basavaraj Padmashali
DOI: 10.7324/JAPS.2019.90217Pages: 124-128
Anti-diabetic drug, metformin, and the p38 inhibitor (SB203580) reduces internal organs oxidative stress in non-obese type 2 diabetic rats
Nuttikarn Nokkaew, Jantira Sanit, Podsawee Mongkolpathumrat, Siyamon Boontawee, Supanut Ithipruchyabun, Wannapa Plangklang, Punyanuch Adulyaritthikul, Kantapich Kongpol, Sarawut Kumphune
DOI: 10.7324/JAPS.2019.90502Pages: 012-020
3D-QSAR, molecular docking and dynamics simulation of difluorophenol pyridine derivatives as RSK2 inhibitor
Muhammad Arba, Hamzah Azali, Sabarudin Ombe, Alrum Armid, Ida Usman
DOI: 10.7324/JAPS.2019.90601Pages: 001-009
15N-NMR spectroscopic studies and investigation of spectral data property relationships of proton pump inhibitors
Bhanumathi Devi NC, Someswara Rao N., Tamal Ghosh, Alok Mukerjee
DOI: 10.7324/JAPS.2019.90608Pages: 061-066
Identification of polyketide synthase 13 inhibitor: Pharmacophore-based virtual screening and molecular dynamics simulation
Muhammad Arba, Andy-Nur Hidayat, Henny Kasmawati, Yamin Yamin, Ida Usman
DOI: 10.7324/JAPS.2019.90702Pages: 012-017
The effect of metformin and P38 MAPK inhibitor on diabetic bone porosity in non-obese type 2 diabetic rats
Punyanuch Adulyaritthikul, Jantira Sanit, Nuttikarn Nokkaew, Kantapich Kongpol, Podsawee Mongkolpathumrat, Sakarat na Lampang, Catleya Rojviriya, Sarawut Kumphune
DOI: 10.7324/JAPS.2019.90711Pages: 082-090
Isolation of flavonol rhamnosides from Pometia pinnata leaves and investigation of α-glucosidase inhibitory activity of flavonol derivatives
Fadhila Utari, Afrizal Itam, Syafrizayanti Syafrizayanti, Widya Hasvini Putri, Masayuki Ninomiya, Mamoru Koketsu, Kaori Tanaka, Mai Efdi
DOI: 10.7324/JAPS.2019.90808Pages: 053-065
Synthesis, in-vitro antioxidant activity and in-silico prediction of drug-likeness properties of a novel compound: 4-(3,5-Di-tert-butyl- 4-hydroxybenzylidene)-3-methylisoxazol-5(4H)-one
Madhavi Kuchana, Durga Rani Bethapudi, Ragini Katamarajugari Ediga, Yoshitha Sisapuram
DOI: 10.7324/JAPS.2019.90915Pages: 105-110
Synthesis, characterization, and in vitro release of oxytetracycline loaded in pH-responsive CaCO3 nanoparticles
Sherifat Banke Idris, Arifah Abdul Kadir, Faez Firdaus Abdullah Jesse, Siti Zubaidah Ramanoon, Muhammad Abdul Basit, Zainul Amiruddin Zakaria, Md Zuki Abu Bakar Zakaria
DOI: 10.7324/JAPS.2019.91103Pages: 019-027
Believes versus evidence-based regio-orientation in the structure assignment of pyrazolo[1,5-a]pyrimidines
Mosaad Sayed Mohamed, Asmaa Mahmoud Mahmoud
DOI: 10.7324/JAPS.2019.91117Pages: 126-144
Pharmacokinetic drug–drug interaction study between clindamycin and cyclosporin in rabbits
Issam Mohammed Abushammala, Lama Attef El Gussein, Badea Elzaman Zomlot, Kamal Fakher Abushammalleh, Mohammed Mahmoud Taha, Mohammed Yousef Miqdad
DOI: 10.7324/JAPS.2020.102016Pages: 108-111
Isolation, characterization, and cytotoxic studies of secondary metabolites from the leaves of Bauhinia foveolata Dalzell: An endemic tree from the Western Ghats, India
Prasanna V. Habbu, Narayan Miskin1, Venkatrao H. Kulkarni, Pradeep Bhat, Arun Joshi, Anant Bhandarkar, Satish Kulkarni, Sheshagiri R. Dixit, Jaishree Vaijanathappa
DOI: 10.7324/JAPS.2020.103018Pages: 135-148
In silico and in vitro assay of Hexagamavunon-6 analogs, Dibenzilyden-N-Methyl-4-piperidone as antibacterial agents
Tesia Aisyah Rahmania, Ritmaleni Ritmaleni, Erna Prawita Setyowati
DOI: 10.7324/JAPS.2020.103004Pages: 039-043
Growth inhibition of combined treatment of cationic liposome/p53 complexes and cisplatin on human carcinoma cells
Wanlop Weecharangsan, Robert J. Lee
DOI: 10.7324/JAPS.2020.104006Pages: 034-040
Fenugreek (Trigonella foenum-graceum) increases postmenopausal fibroblast-associated COL1A1 and COL3A1 production dominantly through its binding to estrogen receptor beta
Shannaz Nadia Yusharyahya, Kusmarinah Bramono, Andon Hestiantoro, Sarah Qanita Edwar, Indra Kusuma
DOI: 10.7324/JAPS.2020.104004Pages: 022-027
Identification, synthesis, and characterization of β-isomer as process related impurity in production of methocarbamol from guaifenesin
Appala Raju Nemala, Sridevi Chigurupati, Kesavanarayanan Krishnan Selvarajan, Saurabh Bhatia, Sridevi Pingali, Anitha Sadula
DOI: 10.7324/JAPS.2020.10502Pages: 010-015
3D QSAR and docking studies on benzoylsulfonohydrazides as histone acetyltransferase KAT6A inhibitors
MD. Muzaffar-Ur-Rehman, Syed Akbar, Asra Ali Bahazeq
DOI: 10.7324/JAPS.2020.10504Pages: 023-030
Novel aminoalkylated chalcone: Synthesis, biological evaluation, and docking simulation as potent antimalarial agents
Jufrizal Syahri, Hasmalina Nasution, Beta Achromi Nurohmah, Bambang Purwono, Emmy Yuanita
DOI: 10.7324/JAPS.2020.10601Pages: 001-005
Synthesis and biological evaluation of novel substituted pyrrolo[2,3-d]pyrimidines as anticancer agents
Sandip P. Dholakia, Kaushik B. Kanada, Ghanshyam R. Parmar
DOI: 10.7324/JAPS.2020.10602Pages: 006-011
Effect of illness perception on improving asthma symptoms with omega-3 fish oil therapy: Pre-post design
Amelia Lorensia, Mariana Wahyudi, Ananta Yudiarso, Siti Erfina Dwi Kurnia
DOI: 10.7324/JAPS.2020.10609Pages: 062-071
Lapatinib-loaded nanocolloidal polymeric micelles for the efficient treatment of breast cancer
Gunjan Vasant Bonde, Gufran Ajmal, Sarita Kumari Yadav, Pooja Mittal, Brahmeshwar Mishra
DOI: 10.7324/JAPS.2020.10903Pages: 023-029
Insights into the structural features of anticancer 1,6-naphthyridines and pyridopyrimidines as VEGFR-2 inhibitors: 3D-QSAR study
Siddharth J. Modi, Dharti H. Modh, Vithal M. Kulkarni
DOI: 10.7324/JAPS.2020.10101Pages: 001-022
Approaches for synthesis and chemical modification of non-condensed heterocyclic systems based on 1,3,4-oxadiazole ring and their biological activity: A review
Maryan Lelyukh, Marta Martynets, Myroslava Kalytovska, Iryna Drapak, Stefan Harkov, Taras Chaban, Ihor Chaban, Vasyl Matiychuk
DOI: 10.7324/JAPS.2020.1010016Pages: 151-165
In silico studies on pyrazine derivatives for identifying potential inhibitors of PIM-1 kinase
Amena Ali, Abuzer Ali, Mohd. Washid Khan, Abutahir, Ibraheem Husain, Kuldeep Patel, Vivek Asati
DOI: 10.7324/JAPS.2020.10116Pages: 040-049
Study of alterations in pharmacokinetics and pharmacodynamics of Saxagliptin in the presence of Rutin: An interaction study in rats
Naga Raju Kandukoori, Pavani Uppu, Narsimha Reddy Yellu
DOI: 10.7324/JAPS.2020.101111Pages: 081-086
Synthesis and cytotoxic evaluation of novel chromenes and chromene(2,3-d)pyrimidines
Mahmoud N. M. Yousif, Abdel-Rahman B. A. El-Gazzar, Ahmed A. Fayed, May A. El-Manawaty, Nabil M. Yousif
DOI: 10.7324/JAPS.2020.101205Pages: 035-043
Bioguided study of the Antarctic alga Himantothallus grandifolius (A. Geep & E.S.Geep) indicates 13E-Docosenamide as potential antileishmanial agent
Leandro Costa Clementino, Fabio Aurelio Esteves Torres, Angela Maria Arenas Velasquez, Leonardo Villela, Toyota Fujii Mutue, Pio Colepicolo, Marcia A. S. Graminha
DOI: 10.7324/JAPS.2020.101213Pages: 098-103
New benzothiazinone linked 1, 2, 4-triazoles: Design, synthesis, characterization, and evaluation of antitubercular activity
Kannampally Ajmal, Gurubasavaraj V. Pujar, Sethu Arun Kumar, Subhankar P. Mandal, Manisha Singh
DOI: 10.7324/JAPS.2021.110204Pages: 029-038
Cytotoxicity of Quercetin and Quercetin-3-O-rhamnoside of Etlingera elatior (Jack) R.M.Sm. leaves against HeLa Cervical Cancer Cells
Herni Kusriani, Anas Subarnas, Ajeng Diantini, Yoppi Iskandar
DOI: 10.7324/JAPS.2021.110512Pages: 085-090
WRL-68 with the overexpression of CYP3A4 as an in vitro model to assess drug–drug interaction
Nurliana Abd Mutalib, Normala Abd Latip
DOI: 10.7324/JAPS.2021.110408Pages: 057-067
Antibacterial evaluation and molecular properties of pyrazolo[3,4-b] pyridines and thieno[2,3-b]pyridines
Mervat A. Elsherif
DOI: 10.7324/JAPS.2021.110614Pages: 118-124
Growth inhibition of cholic acid-conjugated polyethylenimine 25K/ p53-EGFP complexes on human carcinoma cells
Wanlop Weecharangsan, Nattisa Niyomtham, Boon-ek Yingyongnarongkul, Praneet Opanasopit, Robert J. Lee
DOI: 10.7324/JAPS.2021.110403Pages: 014-021
Micropatterned κ-carrageenan-PVP-PEG hydrogels as a templet for head and neck cancer spheroid culture
Nadia Halib, Zainah Adam, Maznah Mahmud
DOI: 10.7324/JAPS.2021.110503Pages: 015-021
Nephroprotectivity of Coccinia indica leaves against gentamycin-induced nephrotoxicity using in vitro and in vivo models
Neelima Satrasala, Dwarakanadha Reddy Peram, Chandra Sekhar Kothapalli Bannoth
DOI: 10.7324/JAPS.2021.110616Pages: 132-139
Isolation, peroxisome proliferator-activated receptor-gamma transcription, glucose uptake, and molecular docking of tetramethoxyflavonoids from the leaves of Rourea mimosoides (Vahl) Planch.
Che Puteh Osman, Norhafizoh Abdul Somat, Zuriati Zahari, Syahrul Imran, Mohd Ilham Adenan
DOI: 10.7324/JAPS.2021.110802Pages: 010-016
Immunopotentiation of galangal (Alpinia galanga L.) when combined with T-cells against metastatic triple-negative breast cancer, MDA-MB 231
Iffan Alif, Rohmad Yudi Utomo, Faradiba Nur Ahlina, Nadzifa Nugraheni, Dedy Hermansyah, Agung Putra, Edy Meiyanto
DOI: 10.7324/JAPS.2021.1101107Pages: 053–061
Design, synthesis and in silico prediction of drug-likeness properties of new ortho, meta and para-(2-cyano-3-(3,5-di-tert-butyl-4- hydroxyphenyl)acrylamido)benzoic acids
Madhavi Kuchana, Lakshmi Bhavani Kambala
DOI: 10.7324/JAPS.2021.110805Pages: 031-035
Novel glitazone attenuates rotenone-induced toxicity in mouse model of Parkinson’s disease
Ankith B. Shetty, Kamsagara Linganna Krishna, Bommenahally Ravanappa Prashantha Kumar, Hittanahalli Shivakumar Nandini
DOI: 10.7324/JAPS.2021.1101007Pages: 042-049
Prevalence of OCT1 (rs628031) genetic polymorphism in south Indian population
Swathi Swaroopa Borra, Bhavya Chebrolu, Poojitha Thotakura, Sujin Bright Francis Joice, Vasanth Raj Palanimuthu, Sadagoban Gopal Krishnamoorthy, Arun Kanniyappan Parthasarathy
DOI: 10.7324/JAPS.2021.1101006Pages: 035-041
Nanodelivery systems for Alzheimer's disease: Prospects of natural therapeutic agents
Oluwatoyin A. Odeku, Tolulope O. Ajala
DOI: 10.7324/JAPS.2021.1101101Pages: 001-010
Biochemical characterization and ecofriendly field application of the plant growth-promoting rhizobacterium Bacillus amyloliquefaciens MH046937 isolated from Salsola imbricata in Tur Sinai, Egypt
Warda E. Ashour, Moustafa M. Zohair, Ahmed A. El-Beih, Eman R. Hamed, Abeer A. Abd El Aty
DOI: 10.7324/JAPS.2021.120109Pages: 094-105
Analysis of the literature on 3D printing in healthcare with reference to pharmaceuticals using a bibliometric approach
Virendra S. Ligade, Akash Chimegave
DOI: 10.7324/JAPS.2022.120310Pages: 096–102
Preparation and evaluation of novel self-dispersing lipid formulation of nevirapine for oral delivery
Gopalapura Bellaiah Preethi, Hagalavadi Nanjappa Shivakumar, Madalli Ravi Kumar
DOI: 10.7324/JAPS.2022.120313Pages: 123–131
The glucose uptake of type 2 diabetic rats by Sargassum olygocystum extract: In silico and in vivo studies
Muhamad Firdaus, Rahmi Nurdiani , Bachtiar Rivai, Windy Hapsari Hemassonida, Aqilatul Badzliyah, Nur Khasanah Sugiat
DOI: 10.7324/JAPS.2022.120314Pages: 132–139
Phytochemical screening, docking study, and in vitro assessment of cytotoxicity against MCF7 and 3T3 cell lines of Indonesian sea cucumber Stichopus sp.
Teni Ernawati , Minarti Minarti, Galuh Widiyarti, Megawati Megawati, Faiza Maryani
DOI: 10.7324/JAPS.2022.120411Pages: 096-107
Overexpression of soluble recombinant Thermus thermophilus (Tth) DNA polymerase in Escherichia coli BL21(DE3) using an MBP fusion tag as a solubility enhancer
Iman Permana Maksum, Diandra Firdiani Utami, Eva Annisa Nurhakim, Yosua, Sriwidodo, Muhammad Yusuf, Muhammad Fadhlillah, Ryan Adibagus Haryanto
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In vitro antiplasmodial activities of the fractions of Hyrtios reticulatus sponge extract
Mahfur Mahfur, Indah Purwantini, Subagus Wahyuono, Erna Prawita Setyowati
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Impact of Morus alba L. on the expression of drug-metabolizing enzymes and transporters in Caco-2 cells
Waranya Chatuphonprasert, Wipawee Tukum-mee, Jintanaporn Wattanathorn, Kanokwan Jarukamjorn
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